SCHEMBL20525358

SCHEMBL20525358

NC(=O)c1ccc(Cn2ccc3cc(C4CCN(Cc5ccncc5)CC4)cnc32)cc1O

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 1/20 0.42
PARP1 P09874 1/20 0.39
CCR5 P51681 4/20 0.39
SCN9A Q15858 1/20 0.37
SYK P43405 1/20 0.35
CNR1 P21554 1/20 0.35
CNR2 P34972 1/20 0.35
SIGMAR1 Q99720 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20525317 0.92 EGLN1 (0.39) EGLN1CCR5SYKCNR1CNR2
SCHEMBL20525414 0.92 PARP1 (0.42) EGLN1PARP1CCR5SCN9ASIGMAR1
SCHEMBL20525400 0.92 PARP1 (0.41) EGLN1PARP1CCR5CNR1CNR2
SCHEMBL20525454 0.92 SYK (0.42) EGLN1PARP1SYK
SCHEMBL20525469 0.91 PIK3CA (0.42) EGLN1PARP1
SCHEMBL20525424 0.91 EGLN1 (0.38) EGLN1CCR5SYKCNR1CNR2
SCHEMBL20525438 0.90 DRD2 (0.42) EGLN1CCR5SYK
SCHEMBL20525339 0.88 PARP1 (0.41) EGLN1PARP1
SCHEMBL20525460 0.88 PARP1 (0.41) EGLN1PARP1SYK
SCHEMBL20525322 0.86 EGLN1 (0.35) EGLN1CCR5SYKCNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3080125-B1 NOVEL AZAINDOLE DERIVATIVES AS SELECTIVE HISTONE DEACETYLASE (HDAC) INHIBITORS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME CHONG KUN DANG PHARMACEUTICAL CORP (KR) 2018-10-10 EP disclosed