SCHEMBL20526344

SCHEMBL20526344

COc1c(O)c(Cl)c2c(c1OC)C1(OC(=O)c3ccc(C(=O)O)cc31)c1ccc(O)c(Cl)c1O2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMAD3 P84022 1/20 0.41
GNG2 P59768 1/20 0.39
GNB1 P62873 1/20 0.39
GAA P10253 1/20 0.34
PKM P14618 1/20 0.34
HTT P42858 1/20 0.33
TPMT P51580 1/20 0.32
DHFR P00374 2/20 0.32
TDP1 Q9NUW8 4/20 0.32
THRB P10828 3/20 0.32
RECQL P46063 3/20 0.32
MEN1 O00255 3/20 0.32
KMT2A Q03164 3/20 0.32
ALDH1A1 P00352 2/20 0.32
BLM P54132 2/20 0.32
CYP3A4 P08684 1/20 0.32
HPGD P15428 1/20 0.32
TSHR P16473 1/20 0.32
MAPK1 P28482 1/20 0.32
CASP1 P29466 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30929844 0.86 GNG2 (0.55) SMAD3GNG2GNB1HTTDHFR
SCHEMBL2167804 0.85 SMAD3 (0.43) SMAD3GNG2GNB1GAAPKM
SCHEMBL15019692 0.84 GNG2 (0.50) SMAD3GNG2GNB1GAAPKM
SCHEMBL29401708 0.84 GNG2 (0.50) SMAD3GNG2GNB1GAAPKM
SCHEMBL2316418 0.82 GNG2 (0.47) SMAD3GNG2GNB1GAAPKM
SCHEMBL20526266 0.81 SMAD3 (0.49) SMAD3GNG2GNB1GAAPKM
SCHEMBL1682554 0.80 SMAD3 (0.40) SMAD3GNG2GNB1TDP1THRB
SCHEMBL29838713 0.79 MEN1 (0.39) GNG2GNB1GAAPKMHTT
SCHEMBL29353753 0.79 MEN1 (0.39) GNG2GNB1GAAPKMHTT
SCHEMBL16118 0.79 MEN1 (0.39) GNG2GNB1GAAPKMHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2687513-B1 DRUGS FOR INHIBITING AGGREGATION OF PROTEINS INVOLVED IN DISEASES LINKED TO PROTEIN AGGREGATION AND/OR NEURODEGENERATIVE DISEASES UNIV MUENCHEN LUDWIG MAXIMILIANS (DE) 2020-12-02 EP disclosed
EP-3385699-A1 OPTOFLUIDIC DEVICE AND METHOD FOR DETECTING CIRCULATING TUMOUR CELLS Universitat Rovira i Virgili (ES) 2018-10-10 EP disclosed