SCHEMBL2052765

SCHEMBL2052765

Fc1ccc(F)c(-c2[c]cccc2C(F)(F)F)c1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 1/20 0.35
PDE3B Q13370 2/20 0.33
PDE3A Q14432 2/20 0.33
HSD11B1 P28845 2/20 0.33
PTPN1 P18031 1/20 0.33
IDO1 P14902 2/20 0.32
TRPA1 O75762 1/20 0.31
PDK2 Q15119 1/20 0.31
CYP11B2 P19099 1/20 0.31
GPR3 P46089 1/20 0.30
AR P10275 2/20 0.30
SLC22A12 Q96S37 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2053791 0.87 HSD11B1 (0.35) CHRM5PDE3BPDE3AHSD11B1IDO1
SCHEMBL2437985 0.81 HSD11B1 (0.38) HSD11B1TRPA1PDK2GPR3AR
SCHEMBL17514845 0.81 HSD11B1 (0.48) HSD11B1TRPA1AR
SCHEMBL17514962 0.78 HSD11B1 (0.48) HSD11B1TRPA1PDK2
SCHEMBL2050214 0.77 PTPN1 (0.34) HSD11B1PTPN1
SCHEMBL2049864 0.77 S1PR2 (0.37) PTPN1
SCHEMBL17514475 0.77
SCHEMBL2433532 0.76 NR1H2 (0.35) CYP11B2AR
SCHEMBL3636361 0.75 HSD11B1 (0.42) HSD11B1TRPA1PDK2AR
SCHEMBL2049471 0.75 HSD11B1 (0.46) PDE3BPDE3AHSD11B1TRPA1PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013182433-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-12-12 WO disclosed
EP-2547687-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-01-23 EP disclosed
EP-2513067-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2012-10-24 EP disclosed
WO-2011073145-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2011-06-23 WO disclosed