SCHEMBL2053791

SCHEMBL2053791

Fc1ccc(-c2[c]cccc2C(F)(F)F)c(F)c1

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 3/20 0.35
AKR1C3 P42330 1/20 0.33
AKR1C2 P52895 1/20 0.33
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
AR P10275 5/20 0.33
ABCC8 Q09428 1/20 0.33
KCNJ11 Q14654 1/20 0.33
P2RX7 Q99572 1/20 0.32
ALOX5AP P20292 1/20 0.32
FEN1 P39748 1/20 0.32
CHRM5 P08912 1/20 0.32
TRPA1 O75762 2/20 0.32
IDO1 P14902 2/20 0.32
PDK2 Q15119 1/20 0.31
GLA P06280 1/20 0.31
POLB P06746 1/20 0.31
GAA P10253 1/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2052765 0.87 CHRM5 (0.35) HSD11B1PDE3BPDE3AARCHRM5
SCHEMBL17514845 0.84 HSD11B1 (0.48) HSD11B1ARP2RX7TRPA1
SCHEMBL17514962 0.84 HSD11B1 (0.48) HSD11B1AKR1C3AKR1C2ALOX5APFEN1
SCHEMBL2437985 0.81 HSD11B1 (0.38) HSD11B1AKR1C3AKR1C2ARTRPA1
SCHEMBL436100 0.81 NFE2L2 (0.36) IDO1
SCHEMBL17514475 0.80
SCHEMBL16720359 0.77 ALDH1A1 (0.40)
SCHEMBL434297 0.77 HSD11B1 (0.36) HSD11B1P2RX7GAA
SCHEMBL2050049 0.77 MAPK14 (0.34) POLB
SCHEMBL2433532 0.76 NR1H2 (0.35) ARGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013182433-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-12-12 WO disclosed
EP-2547687-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-01-23 EP disclosed
EP-2513067-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2012-10-24 EP disclosed
WO-2011113820-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2011-09-22 WO disclosed
WO-2011073145-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2011-06-23 WO disclosed