SCHEMBL20535547

SCHEMBL20535547

CCOC(=O)c1[nH]c2cc(Br)ccc2c1F

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 7/20 0.50
MAPT P10636 4/20 0.50
GABRA1 P14867 1/20 0.47
GABRB1 P18505 1/20 0.47
GABRA3 P34903 1/20 0.47
GABRB2 P47870 1/20 0.47
KDM4E B2RXH2 3/20 0.47
ALDH1A1 P00352 3/20 0.47
NPC1 O15118 2/20 0.47
GAA P10253 2/20 0.47
RAB9A P51151 2/20 0.47
TP53 P04637 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
HPGD P15428 2/20 0.46
NPSR1 Q6W5P4 1/20 0.46
PDE3B Q13370 1/20 0.45
PDE3A Q14432 1/20 0.45
LMNA P02545 1/20 0.45
GPR17 Q13304 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7921819 0.89 ALDH1A1 (0.53) MAPTGABRA1GABRB1GABRA3GABRB2
SCHEMBL24074581 0.86 ALDH1A1 (0.58) ALOX15MAPTGABRA1GABRB1GABRA3
SCHEMBL8795754 0.85 ALOX15 (0.61) ALOX15MAPT
SCHEMBL24113129 0.85 MAPT (0.48) ALOX15MAPTKDM4EALDH1A1NPC1
SCHEMBL28477589 0.84 KDM4E (0.64) ALOX15MAPTGABRA1GABRB1GABRA3
SCHEMBL30071216 0.82 ALOX15 (0.54) ALOX15MAPTKDM4EALDH1A1NPC1
SCHEMBL20494685 0.82 ALOX15 (0.54) ALOX15MAPTKDM4EALDH1A1NPC1
SCHEMBL28640836 0.82 ALOX15 (0.73) ALOX15MAPTGABRA1GABRB1GABRA3
SCHEMBL29955347 0.82 ALOX15 (0.73) ALOX15MAPTGABRA1GABRB1GABRA3
SCHEMBL21822255 0.81 ALOX15 (0.47) ALOX15MAPTKDM4EALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250243202-A1 Compounds Useful as RET Inhibitors CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2025-07-31 US disclosed
CN-115785100-B Compounds useful as RET inhibitors 癌症研究科技有限公司 2025-01-07 CN disclosed
US-20240132504-A1 Compounds Useful as RET Inhibitors CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2024-04-25 US disclosed
US-11680068-B2 Compounds useful as RET inhibitors CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2023-06-20 US disclosed
CN-115785100-A Compounds useful as RET inhibitors 癌症研究科技有限公司 2023-03-14 CN disclosed
EP-4105219-A1 PYRAZOLOPYRIMIDINE COMPOUNDS USEFUL AS RET INHIBITORS Cancer Research Technology Limited (GB) 2022-12-21 EP disclosed
US-20220348585-A1 Compounds Useful as RET Inhibitors CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2022-11-03 US disclosed
CN-110506043-B Compounds useful as RET inhibitors 癌症研究科技有限公司 2022-11-01 CN disclosed
US-11352361-B2 Compounds useful as RET inhibitors CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2022-06-07 US disclosed
EP-3609898-B1 COMPOUNDS USEFUL AS RET INHIBITORS CANCER RESEARCH TECH LTD (GB) 2022-06-01 EP disclosed
US-20200157107-A1 Compounds Useful as RET Inhibitors CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2020-05-21 US disclosed
EP-3609898-A1 COMPOUNDS USEFUL AS RET INHIBITORS Cancer Research Technology Limited (GB) 2020-02-19 EP disclosed
WO-2018189553-A1 COMPOUNDS USEFUL AS RET INHIBITORS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2018-10-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250243202-A1 Compounds Useful as RET Inhibitors RET, BCR, REL ALOX15 3511/4885MAPT 3607/4885GABRA1 2548/4885
US-20220348585-A1 Compounds Useful as RET Inhibitors RET, BCR, REL ALOX15 3511/4885MAPT 3607/4885GABRA1 2548/4885
US-11352361-B2 Compounds useful as RET inhibitors RET, BCR, REL ALOX15 3511/4885MAPT 3607/4885GABRA1 2548/4885
US-20200157107-A1 Compounds Useful as RET Inhibitors RET, BCR, REL ALOX15 3511/4885MAPT 3607/4885GABRA1 2548/4885
US-20240132504-A1 Compounds Useful as RET Inhibitors RET, BCR, REL ALOX15 3511/4885MAPT 3607/4885GABRA1 2548/4885
US-11680068-B2 Compounds useful as RET inhibitors RET, BCR, REL ALOX15 3511/4885MAPT 3607/4885GABRA1 2548/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.