SCHEMBL20537804

SCHEMBL20537804

COc1cc(/C=C/c2cc(OC)c(OC)c(OC)c2)ccc1NC(=O)/C=C/c1ccc([N+](=O)[O-])cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.68
KRAS P01116 2/20 0.62
TRPV1 Q8NER1 1/20 0.60
ALDH1A1 P00352 5/20 0.59
GLA P06280 1/20 0.59
MAPT P10636 4/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
KMT2A Q03164 3/20 0.58
CYP3A4 P08684 2/20 0.58
CYP2C19 P33261 2/20 0.58
MEN1 O00255 2/20 0.58
CYP19A1 P11511 1/20 0.56
NPC1 O15118 1/20 0.55
RAB9A P51151 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
LMNA P02545 2/20 0.54
KDM4E B2RXH2 2/20 0.54
GAA P10253 1/20 0.54
HPGD P15428 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20537805 1.00 PTGS2 (0.68) PTGS2KRASTRPV1ALDH1A1GLA
SCHEMBL20538038 0.93 PTGS2 (0.64) PTGS2KRASTRPV1ALDH1A1GLA
SCHEMBL20538041 0.93 PTGS2 (0.64) PTGS2KRASTRPV1ALDH1A1GLA
SCHEMBL20537790 0.93 PTGS2 (0.67) PTGS2KRASTRPV1ALDH1A1MAPT
SCHEMBL20537791 0.93 PTGS2 (0.67) PTGS2KRASTRPV1ALDH1A1MAPT
SCHEMBL20538326 0.93 PTGS2 (0.70) PTGS2KRASTRPV1ALDH1A1MAPT
SCHEMBL20538324 0.93 PTGS2 (0.70) PTGS2KRASTRPV1ALDH1A1MAPT
SCHEMBL20538089 0.91 TRPV1 (0.74) PTGS2KRASTRPV1ALDH1A1GLA
SCHEMBL20538500 0.90 TUBB4A (0.63) TRPV1ALDH1A1MAPTSMN1; SMN2KMT2A
SCHEMBL20538498 0.90 TUBB4A (0.63) TRPV1ALDH1A1MAPTSMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3183230-B1 N-((3,4,5-TRIMETHOXYSTYRYL)ARYL)CINNAMAMIDE COMPOUNDS AS POTENTIAL ANTICANCER AGENTS AND PROCESS FOR THE PREPARATION THEREOF COUNCIL SCIENT IND RES (IN) 2018-10-24 EP claimed