SCHEMBL2054526

SCHEMBL2054526

Cc1ccc(CCCCN(C[C@H](O)c2ccc(O)c(O)c2)C[C@H](O)c2ccc(O)c(NC=O)c2)cc1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 18/20 0.49
ADRB1 P08588 10/20 0.47
ADRB3 P13945 8/20 0.47
DRD2 P14416 2/20 0.43
PGR P06401 1/20 0.43
SLC6A4 P31645 1/20 0.43
ADRA1A P35348 1/20 0.43
PTGS2 P35354 1/20 0.43
SLC6A3 Q01959 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
TSHR P16473 1/20 0.43
MAPK1 P28482 1/20 0.43
CYP2C19 P33261 1/20 0.43
DRD3 P35462 1/20 0.43
IGF1R P08069 1/20 0.43
ALOX15 P16050 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2054463 0.87 ADRB2 (0.51) ADRB2ADRB1ADRB3DRD2PGR
Acetic Acid SCHEMBL967644 0.85 ADRB2 (0.49) ADRB2ADRB1ADRB3DRD2PGR
Acetic Acid SCHEMBL967642 0.85 ADRB2 (0.49) ADRB2ADRB1ADRB3DRD2PGR
SCHEMBL2056281 0.81 ADRB2 (0.65) ADRB2ADRB1ADRB3DRD2PGR
SCHEMBL12920490 0.76 SCNN1A (0.38) ADRB2ADRB1ADRB3DRD2PGR
SCHEMBL13042337 0.74 ADRB3 (0.57) ADRB2ADRB1ADRB3DRD2PGR
SCHEMBL11819755 0.74 ADRB2 (0.65) ADRB2ADRB1ADRB3DRD2PGR
SCHEMBL3979708 0.72 ADRB2 (0.53) ADRB2ADRB1ADRB3DRD2PGR
SCHEMBL13807382 0.72 ADRB2 (0.53) ADRB2ADRB1ADRB3DRD2PGR
SCHEMBL10036716 0.71 ADRB2 (0.79) ADRB2ADRB1ADRB3DRD2PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8163758-B2 Phenyl substituted pyrazinoylguanidine sodium channel blockers possessing beta agonist activity PARION SCIENCES, INC. (US) 2012-04-24 US disclosed