SCHEMBL2054779

SCHEMBL2054779

CCC(NC(=O)c1ccc(C(F)(F)F)nc1C)c1nnc(S(=O)(=O)CC2CC2)n1C

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 2/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
RORC P51449 8/20 0.37
LMNA P02545 1/20 0.37
CYP2C9 P11712 1/20 0.36
GAA P10253 1/20 0.36
CTPS1 P17812 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2054776 0.93 NPC1 (0.38) KCNK3NPC1RAB9ARORCLMNA
SCHEMBL8251813 0.92 NPC1 (0.38) KCNK3NPC1RAB9ARORCLMNA
SCHEMBL2097455 0.92 NPC1 (0.38) KCNK3NPC1RAB9ARORCLMNA
SCHEMBL2054772 0.92 NPC1 (0.37) KCNK3NPC1RAB9ARORCLMNA
SCHEMBL2054777 0.88 KCNK3 (0.39) KCNK3NPC1RAB9ARORCLMNA
SCHEMBL2054774 0.73 RORC (0.32) RORC
SCHEMBL2054773 0.72 SLC6A9 (0.42)
SCHEMBL2054775 0.71 NPC1 (0.42) KCNK3NPC1RAB9ALMNAGAA
SCHEMBL2054766 0.71 NPC1 (0.41) NPC1RAB9ALMNAGAA
SCHEMBL5431669 0.69 NPC1 (0.56) NPC1RAB9ALMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8163956-B2 Inhibitors of GLYT1 transporters MERCK SHARP & DOHME CORP. (US) 2012-04-24 US disclosed