SCHEMBL20558458

SCHEMBL20558458

CC(N)c1c(F)cccc1Br

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.35
MAOB P27338 1/20 0.35
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33
PDE2A O00408 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
NFKB1 P19838 1/20 0.31
PNMT P11086 1/20 0.31
HTT P42858 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
GLA P06280 1/20 0.31
SLC6A2 P23975 2/20 0.30
TAAR1 Q96RJ0 2/20 0.30
SLC6A4 P31645 1/20 0.30
SLC6A3 Q01959 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16356139 0.84 HTR2A (0.39) MAOAHTR2AHTR2CCES2CES1
SCHEMBL1239996 0.84 HTR2A (0.39) MAOAHTR2AHTR2CCES2CES1
SCHEMBL16908267 0.84 HTR2A (0.39) MAOAHTR2AHTR2CCES2CES1
SCHEMBL12986654 0.83 CES2 (0.35) HTR2CCES2CES1CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL20445854 0.82 ALDH1A1 (0.39) MAOAHTR2AHTR2CCES2CES1
Hydrochloric Acid SCHEMBL20445855 0.82 ALDH1A1 (0.39) MAOAHTR2AHTR2CCES2CES1
Hydrochloric Acid SCHEMBL16321559 0.82 ALDH1A1 (0.39) MAOAHTR2AHTR2CCES2CES1
SCHEMBL6745071 0.79 CES2 (0.41) MAOBCES2CES1HTTALDH1A1
SCHEMBL30266772 0.76 CES2 (0.36) MAOBCES2CES1HTT
SCHEMBL2268624 0.76 CES2 (0.36) MAOBCES2CES1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018205948-A1 COMPOUNDS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2018-11-15 WO disclosed