SCHEMBL2056695

SCHEMBL2056695

Cc1cn([C@H]2CC(O)[C@@H](C)O2)c(=O)[nH]c1=O

nearest known ligand 0.72

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TK1 P04183 5/20 0.72
DHFR P00374 1/20 0.57
POLB P06746 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14682231 1.00 TK1 (0.72) TK1DHFRPOLB
SCHEMBL2056693 1.00 TK1 (0.72) TK1DHFRPOLB
Iodide SCHEMBL8583592 0.99 TK1 (0.70) TK1DHFRPOLB
Hydrochloric Acid SCHEMBL8585203 0.99 TK1 (0.70) TK1DHFRPOLB
SCHEMBL12718422 0.93 TK1 (0.67) TK1DHFRPOLB
SCHEMBL17236359 0.93 TK1 (0.67) TK1DHFRPOLB
SCHEMBL12718420 0.92 TK1 (0.66) TK1DHFR
SCHEMBL14590480 0.87 TK1 (0.59) TK1DHFR
SCHEMBL7200634 0.86 TK1 (0.69) TK1DHFRPOLB
SCHEMBL4348630 0.86 TK1 (0.69) TK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 68 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1131270-B1 PROCESS FOR CONVERTING AN ALCOHOL TO THE CORRESPONDING FLUORIDE 3M INNOVATIVE PROPERTIES CO (US) 2004-04-07 EP claimed
US-6248889-B1 FORMING MIXTURE COMPRISING AT LEAST ONE FLUORINATED, SATURATED ALIPHATIC OR ALICYCLIC SULFONYL FLUORIDE AND AT LEAST ONE PRIMARY OR SECONDARY ALCOHOL, ADDING MOLAR EXCESS OF STRONG, APROTIC, NON-NUCLEOPHILIC HINERED ORGANIC BASE 3M INNOVATIVE PROPERTIES COMPANY 2001-06-19 US claimed
EP-0360820-B1 OLIGOBIPYRIDINE LIGANDS, PROCESS FOR OBTAINING THEM AND APPLICATION AS COMPLEXING AGENTS CIS BIO INTERNATIONAL (FR) 1992-08-19 EP claimed
EP-0360820-A1 OLIGOBIPYRIDINE LIGANDS, PROCESS FOR OBTAINING THEM AND APPLICATION AS COMPLEXING AGENTS. ORIS SA (FR) 1990-04-04 EP claimed
WO-1988008419-A1 OLIGOBIPYRIDINE LIGANDS, PROCESS FOR OBTAINING THEM AND APPLICATION AS COMPLEXING AGENTS COMPAGNIE ORIS INDUSTRIE S.A. (FR) 1988-11-03 WO claimed
EP-4745237-A1 RNAI AGENT FOR INHIBITING EXPRESSION OF KETOHEXOKINASE AND USE THEREOF YUN HO BIO CO., LTD (CN) 2026-05-20 EP disclosed
EP-4722363-A1 RNAI AGENT FOR INHIBITING ANGPTL3 EXPRESSION AND USE THEREOF YUN HO BIO CO., LTD (CN) 2026-04-08 EP disclosed
EP-4634385-A2 RNAI CONSTRUCTS FOR INHIBITING TTR EXPRESSION AND METHODS OF USE THEREOF AMGEN INC. (US) 2025-10-22 EP disclosed
US-20250320502-A1 RNAI CONSTRUCTS FOR INHIBITING PNPLA3 EXPRESSION AND METHODS OF USE THEREOF AMGEN INC. (US) 2025-10-16 US disclosed
US-20250313834-A1 RNAI CONSTRUCTS FOR INHIBITING SCAP EXPRESSION AND METHODS OF USE THEREOF AMGEN INC. (US) 2025-10-09 US disclosed
US-20250207138-A1 RNAI CONSTRUCTS FOR INHIBITING PNPLA3 EXPRESSION AND METHODS OF USE THEREOF AMGEN INC. (US) 2025-06-26 US disclosed
EP-4562152-A2 RNAI CONSTRUCTS AND METHODS FOR INHIBITING FAM13A EXPRESSION Amgen Inc. (US) 2025-06-04 EP disclosed
US-5910406-A HYBRIDIZING ON SOLID SUPPORT TEPNEL MEDICAL LIMITED (GB) 1999-06-08 US disclosed
US-5777092-A Heteroatomic oligonucleoside linkages ISIS PHARMACEUTICALS, INC. (US) 1998-07-07 US disclosed
EP-0767668-A4 POLYNUCLEOSIDE CHAIN HAVING MULTIPLE NUCLEOSIDES, THE NUCLEOSIDES COUPLED BY GUANIDYL LINKAGES UNIV CALIFORNIA (US) 1998-04-08 EP disclosed
EP-0767668-A1 POLYNUCLEOSIDE CHAIN HAVING MULTIPLE NUCLEOSIDES, THE NUCLEOSIDES COUPLED BY GUANIDYL LINKAGES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1997-04-16 EP disclosed
EP-0348458-B1 DNA MOLECULES STABILIZED BY MODIFICATIONS OF THE 3'-TERMINAL PHOSPHODIESTER LINKAGE AND THEIR USE AS NUCLEIC ACID PROBES AND AS THERAPEUTIC AGENTS TO BLOCK THE EXPRESSION OF SPECIFICALLY TARGETED GENES UNIV IOWA RES FOUND (US) 1997-04-09 EP disclosed
US-5491133-A CONTACTING EUKARYOTIC CELL IN VITRO WITH OLIGODEOXYNUCLEOTIDE WHICH HAS COMPLEMENTARITY FOR AND IS HYBRIDIZABLE TO SPECIFED MESSENGER RNA REGION AND HAS MODIFIED PHOSPHODIESTER LINKAGE RESISTANT TO EXONUCLEASE DEGRADATION UNIVERSITY OF IOWA RESEARCH FOUNDATION (US) 1996-02-13 US disclosed
WO-1996000575-A1 POLYNUCLEOSIDE CHAIN HAVING MULTIPLE NUCLEOSIDES, THE NUCLEOSIDES COUPLED BY GUANIDYL LINKAGES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1996-01-11 WO disclosed
WO-1989005358-A1 DNA AND RNA MOLECULES STABILIZED BY MODIFICATIONS OF THE 3'-TERMINAL PHOSPHODIESTER LINKAGE AND THEIR USE AS NUCLEIC ACID PROBES AND AS THERAPEUTIC AGENTS TO BLOCK THE EXPRESSION OF SPECIFICALLY TARGETED GENES UNIVERSITY OF IOWA RESEARCH FOUNDATION (US) 1989-06-15 WO disclosed