SCHEMBL20567883

SCHEMBL20567883

CN(C)CCNC(=O)c1ccc([N+](=O)[O-])cc1C(F)(F)F

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.53
MAPT P10636 5/20 0.53
MEN1 O00255 3/20 0.53
KMT2A Q03164 3/20 0.53
LMNA P02545 3/20 0.52
HTT P42858 6/20 0.51
POLB P06746 3/20 0.51
MAPK1 P28482 1/20 0.51
GAA P10253 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.48
TP53 P04637 1/20 0.47
RORC P51449 1/20 0.45
TMEM97 Q5BJF2 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
KDM4E B2RXH2 2/20 0.43
CYP1A2 P05177 1/20 0.43
ESRRG P62508 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31203036 0.83 HTT (0.67) ALDH1A1MAPTLMNAHTTPOLB
SCHEMBL26757977 0.81 HTT (0.56) ALDH1A1MAPTMEN1KMT2ALMNA
SCHEMBL20568584 0.80 SMN1; SMN2 (0.52) ALDH1A1KMT2ALMNAHTTPOLB
SCHEMBL6111089 0.80 MCHR1 (0.53) ALDH1A1MAPTMEN1KMT2AHTT
SCHEMBL7460757 0.79 CYP1A2 (0.64) MAPTMEN1KMT2ALMNAHTT
SCHEMBL5713303 0.79 HTT (0.54) ALDH1A1MAPTMEN1KMT2ALMNA
SCHEMBL18770223 0.78 HTT (0.53) ALDH1A1MAPTMEN1KMT2ALMNA
SCHEMBL7476700 0.77 HTT (0.49) ALDH1A1MAPTMEN1KMT2ALMNA
SCHEMBL16045437 0.77 L3MBTL1 (0.60) ALDH1A1MAPTMEN1KMT2ALMNA
SCHEMBL17687389 0.77 GAA (0.55) ALDH1A1MAPTKMT2ALMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112601752-A Novel inhibitors of MAP4K1 伊克诺斯科学公司 2021-04-02 CN disclosed
EP-3630778-A1 NOVEL INHIBITORS OF MAP4K1 Ichnos Sciences SA (CH) 2020-04-08 EP disclosed
WO-2018215668-A1 NOVEL INHIBITORS OF MAP4K1 GLENMARK PHARMACEUTICALS S.A. (CH) 2018-11-29 WO disclosed