SCHEMBL20567977

SCHEMBL20567977

CC(C)NCc1cc([N+](=O)[O-])cc(C(F)(F)F)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.40
TSHR P16473 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
MAPK1 P28482 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
RECQL P46063 1/20 0.38
P2RX1 P51575 2/20 0.38
TDO2 P48775 1/20 0.38
CETP P11597 1/20 0.38
PIN1 Q13526 2/20 0.38
MEN1 O00255 1/20 0.38
PKM P14618 1/20 0.38
KMT2A Q03164 1/20 0.38
IDO1 P14902 1/20 0.37
ALDH1A1 P00352 2/20 0.37
HPGD P15428 1/20 0.37
ALOX15 P16050 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14569541 0.81 IDO1 (0.47) IDO1ALDH1A1LMNA
SCHEMBL4520546 0.79 TSHR (0.53) CYP3A4TSHRTDP1MAPK1L3MBTL1
SCHEMBL26017464 0.79 L3MBTL1 (0.38) CYP3A4TSHRTDP1MAPK1L3MBTL1
SCHEMBL25077871 0.79 CYP3A4 (0.45) CYP3A4TSHRTDP1MAPK1P2RX1
SCHEMBL20568864 0.78 L3MBTL1 (0.43) CYP3A4L3MBTL1P2RX1CETPPIN1
SCHEMBL25771219 0.77 L3MBTL1 (0.37) CYP3A4TSHRTDP1MAPK1L3MBTL1
SCHEMBL4975333 0.76 IDO1 (0.43) CYP3A4TSHRTDP1MAPK1P2RX1
SCHEMBL14493293 0.75 CYP3A4 (0.43) CYP3A4TSHRTDP1MAPK1L3MBTL1
SCHEMBL131155 0.75 ALDH1A1 (0.43) CYP3A4TSHRTDP1MAPK1L3MBTL1
SCHEMBL15542723 0.75 ALDH1A1 (0.43) CYP3A4TSHRTDP1MAPK1P2RX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112601752-A Novel inhibitors of MAP4K1 伊克诺斯科学公司 2021-04-02 CN disclosed
EP-3630778-A1 NOVEL INHIBITORS OF MAP4K1 Ichnos Sciences SA (CH) 2020-04-08 EP disclosed
WO-2018215668-A1 NOVEL INHIBITORS OF MAP4K1 GLENMARK PHARMACEUTICALS S.A. (CH) 2018-11-29 WO disclosed