SCHEMBL20568968

SCHEMBL20568968

CN(C)CCN(C)c1cc(N(C(=O)O)C(=O)O)cc(C(F)(F)F)c1

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 7/20 0.43
BRAF P15056 5/20 0.37
CCR2 P41597 6/20 0.36
ABL1 P00519 1/20 0.35
MCHR1 Q99705 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12398713 0.82 TACR1 (0.43) TACR1BRAFABL1MCHR1
SCHEMBL10104262 0.76 NOS1 (0.45) TACR1BRAFABL1MCHR1
SCHEMBL2201726 0.75 NOS1 (0.39) TACR1BRAFABL1
SCHEMBL15131546 0.74 TEK (0.44) TACR1CCR2
SCHEMBL24781287 0.74 NOS1 (0.41) TACR1CCR2
Hydrochloric Acid SCHEMBL15122987 0.73 TEK (0.43) TACR1CCR2
SCHEMBL13130561 0.73 TACR1 (0.39) TACR1BRAFCCR2
SCHEMBL18794873 0.71 TACR1 (0.52) TACR1
SCHEMBL20568892 0.71 NOTUM (0.46) TACR1
SCHEMBL15397669 0.69 TACR1 (0.59) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3630778-A1 NOVEL INHIBITORS OF MAP4K1 Ichnos Sciences SA (CH) 2020-04-08 EP disclosed
WO-2018215668-A1 NOVEL INHIBITORS OF MAP4K1 GLENMARK PHARMACEUTICALS S.A. (CH) 2018-11-29 WO disclosed