SCHEMBL20570795

SCHEMBL20570795

N#Cc1c(-c2ccccc2)nc(-c2cccnc2)[nH]c1=O

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 5/20 0.77
ALDH1A1 P00352 3/20 0.77
CYP1A2 P05177 1/20 0.77
CYP2C9 P11712 1/20 0.77
KMT2A Q03164 3/20 0.67
MEN1 O00255 2/20 0.67
XDH P47989 1/20 0.59
RXFP1 Q9HBX9 2/20 0.59
PPARG P37231 1/20 0.59
NCOR2 Q9Y618 1/20 0.59
ADORA2A P29274 3/20 0.58
ADORA1 P30542 3/20 0.58
HTT P42858 2/20 0.57
NPSR1 Q6W5P4 1/20 0.57
ADORA2B P29275 1/20 0.54
POLB P06746 1/20 0.52
MAPT P10636 1/20 0.51
KDM4C Q9H3R0 1/20 0.51
KDM4E B2RXH2 1/20 0.51
ACMSD Q8TDX5 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20570670 0.88 HPGD (0.79) HPGDALDH1A1CYP1A2CYP2C9KMT2A
SCHEMBL19665221 0.87 HPGD (1.00) HPGDALDH1A1CYP1A2CYP2C9KMT2A
SCHEMBL20571237 0.82 MAPT (0.56) HPGDALDH1A1CYP1A2CYP2C9KMT2A
SCHEMBL20570664 0.81 HPGD (0.51) HPGDALDH1A1CYP1A2CYP2C9KMT2A
SCHEMBL20569921 0.81 HPGD (0.51) HPGDALDH1A1CYP1A2CYP2C9KMT2A
SCHEMBL20570559 0.81 HPGD (0.76) HPGDALDH1A1CYP1A2CYP2C9KMT2A
SCHEMBL20569911 0.81 HPGD (0.50) HPGDALDH1A1CYP1A2CYP2C9KMT2A
SCHEMBL20569842 0.80 HPGD (0.52) HPGDALDH1A1CYP1A2CYP2C9KMT2A
SCHEMBL20571335 0.80 CYP2C9 (0.55) HPGDALDH1A1CYP1A2CYP2C9KMT2A
SCHEMBL20571330 0.79 ALDH1A1 (0.72) HPGDALDH1A1CYP1A2CYP2C9KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3883577-B1 COMPOSITIONS AND METHODS OF MODULATING SHORT-CHAIN DEHYDROGENASE ACTIVITY UNIV CASE WESTERN RESERVE (US) 2026-04-08 EP disclosed
US-20250304597-A1 COMPOSITIONS AND METHODS OF MODULATING SHORT-CHAIN DEHYDROGENASE ACTIVITY BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM 2025-10-02 US disclosed
US-12336982-B2 Compositions and methods of modulating short-chain dehydrogenase activity RODEO THERAPEUTICS CORPORATION (US) 2025-06-24 US disclosed
CN-113507931-B Compositions and methods for modulating short-chain dehydrogenase activity 卡斯西部储备大学 2025-05-27 CN disclosed
US-20250161277-A1 COMPOSITIONS AND METHODS OF MODULATING SHORT-CHAIN DEHYDROGENASE ACTIVITY BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM 2025-05-22 US disclosed
US-20240043440-A1 COMPOSITIONS AND METHODS OF MODULATING SHORT-CHAIN DEHYDROGENASE ACTIVITY BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM 2024-02-08 US disclosed
US-20230039604-A1 COMPOSITIONS AND METHODS OF MODULATING SHORT-CHAIN DEHYDROGENASE ACTIVITY RODEO THERAPEUTICS CORPORATION 2023-02-09 US disclosed
CN-113507931-A Compositions and methods for modulating short-chain dehydrogenase activity 卡斯西部储备大学 2021-10-15 CN disclosed
US-20210317132-A1 COMPOSITIONS AND METHODS OF MODULATING SHORT-CHAIN DEHYDROGENASE ACTIVITY NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2021-10-14 US disclosed
US-20210317132-A1 COMPOSITIONS AND METHODS OF MODULATING SHORT-CHAIN DEHYDROGENASE ACTIVITY NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2021-10-14 US disclosed
EP-3883577-A1 COMPOSITIONS AND METHODS OF MODULATING SHORT-CHAIN DEHYDROGENASE ACTIVITY CASE WESTERN RESERVE UNIVERSITY (US) 2021-09-29 EP disclosed
CN-111132982-A Compositions and methods for modulating short-chain dehydrogenase activity 卡斯西部储备大学 2020-05-08 CN disclosed
EP-3630773-A1 COMPOSITIONS AND METHODS OF MODULATING SHORT-CHAIN DEHYDROGENASE ACTIVITY Case Western Reserve University (US) 2020-04-08 EP disclosed
WO-2018218251-A1 COMPOSITIONS AND METHODS OF MODULATING SHORT-CHAIN DEHYDROGENASE ACTIVITY CASE WESTERN RESERVE UNIVERSITY (US) 2018-11-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250304597-A1 COMPOSITIONS AND METHODS OF MODULATING SHORT-CHAIN DEHYDROGENASE ACTIVITY HPGD, GCDH, HPGDS HPGD 1/4885ALDH1A1 126/4885CYP1A2 463/4885
US-20210317132-A1 COMPOSITIONS AND METHODS OF MODULATING SHORT-CHAIN DEHYDROGENASE ACTIVITY HPGD, GCDH, HPGDS HPGD 1/4885ALDH1A1 126/4885CYP1A2 463/4885
US-20250161277-A1 COMPOSITIONS AND METHODS OF MODULATING SHORT-CHAIN DEHYDROGENASE ACTIVITY HPGD, GCDH, HPGDS HPGD 1/4885ALDH1A1 126/4885CYP1A2 463/4885
US-20240043440-A1 COMPOSITIONS AND METHODS OF MODULATING SHORT-CHAIN DEHYDROGENASE ACTIVITY HPGD, GCDH, HPGDS HPGD 1/4885ALDH1A1 126/4885CYP1A2 463/4885
US-12336982-B2 Compositions and methods of modulating short-chain dehydrogenase activity HPGD, GCDH, HPGDS HPGD 1/4885ALDH1A1 126/4885CYP1A2 463/4885
US-20230039604-A1 COMPOSITIONS AND METHODS OF MODULATING SHORT-CHAIN DEHYDROGENASE ACTIVITY HPGD, GCDH, HPGDS HPGD 1/4885ALDH1A1 126/4885CYP1A2 463/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.