SCHEMBL20573191

SCHEMBL20573191

Cc1[nH]c2ncc(F)cc2c1C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AGBL2 Q5U5Z8 1/20 0.40
PADI4 Q9UM07 4/20 0.38
DHODH Q02127 8/20 0.37
BRD4 O60885 1/20 0.37
HCAR2 Q8TDS4 1/20 0.35
DHFR P00374 1/20 0.34
ALKBH5 Q6P6C2 1/20 0.34
IDO1 P14902 1/20 0.33
TDO2 P48775 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ASPH Q12797 1/20 0.33
KDM8 Q8N371 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2157057 0.85 NR4A2 (0.47) DHODHBRD4KDM4E
SCHEMBL28757158 0.75 DAO (0.52) PADI4DHODH
SCHEMBL4237180 0.74 PADI4 (0.36) PADI4DHODHHCAR2
SCHEMBL21819026 0.71 AURKA (0.45) DHODHBRD4
SCHEMBL8468860 0.71 TYMS (0.33)
SCHEMBL5857601 0.71 KEAP1 (0.50) KDM4E
SCHEMBL2814713 0.69 AXL (0.47) KDM4EASPHKDM8
SCHEMBL8329308 0.69 MAP4K1 (0.37)
SCHEMBL8329311 0.69 CYP3A4 (0.41) AGBL2KDM4E
SCHEMBL25169884 0.68 PTGS1 (0.55) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2513110-B1 1,7-DIAZACARBAZOLES AND THEIR USE IN THE TREATMENT OF CANCER HOFFMANN LA ROCHE (CH) 2018-12-05 EP disclosed