SCHEMBL20604757

SCHEMBL20604757

CC(C)(C)[Si](C)(C)OC1CCC(n2cc(Br)c3ccccc32)C1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 12/20 0.37
PIM1 P11309 1/20 0.32
MARK3 P27448 1/20 0.32
MAP4K2 Q12851 1/20 0.32
CAMK2B Q13554 1/20 0.32
PIM3 Q86V86 1/20 0.32
PIM2 Q9P1W9 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A3 Q01959 1/20 0.32
CHRM2 P08172 1/20 0.32
CHRM4 P08173 1/20 0.32
CHRM5 P08912 1/20 0.32
CHRM1 P11229 1/20 0.32
CHRM3 P20309 1/20 0.32
MET P08581 1/20 0.31
MAP3K5 Q99683 1/20 0.31
OPRK1 P41145 1/20 0.31
KCNH2 Q12809 1/20 0.31
OPRM1 P35372 1/20 0.31
OPRD1 P41143 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20837926 0.84 HTR3A (0.35) HTR3APIM1MAP4K2MET
SCHEMBL6592321 0.82 HTR3A (0.48) HTR3AOPRK1OPRM1OPRD1OPRL1
SCHEMBL6592314 0.82 HTR3A (0.48) HTR3AOPRK1OPRM1OPRD1OPRL1
SCHEMBL6588979 0.81 HTR3A (0.51) HTR3A
SCHEMBL6588982 0.81 HTR3A (0.51) HTR3A
SCHEMBL20595024 0.79 KDM1A (0.43)
SCHEMBL20657195 0.79 KDM1A (0.43)
SCHEMBL20595251 0.79 KDM1A (0.43)
SCHEMBL23648082 0.75 KDM4E (0.44) CAMK2BOPRK1OPRM1OPRD1OPRL1
SCHEMBL30006023 0.75 KDM4E (0.44) CAMK2BOPRK1OPRM1OPRD1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3423443-A1 CYANO-SUBSTITUTED INDOLE COMPOUNDS AND USES THEREOF AS LSD1 INHIBITORS Novartis AG (CH) 2019-01-09 EP disclosed