SCHEMBL20629916

SCHEMBL20629916

CC(=O)/C(C#N)=C/C(C)(C)N1CCOCC1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ITK Q08881 3/20 0.37
SMN1; SMN2 Q16637 3/20 0.34
BTK Q06187 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
ALDH1A1 P00352 8/20 0.33
MAPT P10636 6/20 0.33
KDM4E B2RXH2 4/20 0.33
KMT2A Q03164 4/20 0.33
USP2 O75604 3/20 0.33
MEN1 O00255 3/20 0.33
GAA P10253 1/20 0.33
THRB P10828 1/20 0.33
HPGD P15428 2/20 0.33
POLB P06746 1/20 0.33
TSHR P16473 2/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20400199 0.88 BTK (0.38) ITKBTKNPC1RAB9AALDH1A1
SCHEMBL20400198 0.88 BTK (0.38) ITKBTKNPC1RAB9AALDH1A1
SCHEMBL20629865 0.86 MAPT (0.38) ITKSMN1; SMN2BTKNPC1RAB9A
SCHEMBL15710719 0.86 MAPT (0.38) ITKSMN1; SMN2BTKNPC1RAB9A
SCHEMBL22370699 0.82 USP2 (0.42) ITKSMN1; SMN2BTKALDH1A1MAPT
SCHEMBL22370702 0.82 USP2 (0.42) ITKSMN1; SMN2BTKALDH1A1MAPT
SCHEMBL20082945 0.82 NPC1 (0.43) ITKSMN1; SMN2BTKNPC1RAB9A
SCHEMBL24991319 0.80 BTK (0.41) BTK
SCHEMBL28976097 0.79 ITK (0.39) ITKBTKNPC1RAB9AALDH1A1
SCHEMBL22439617 0.77 ALDH1A1 (0.38) ITKSMN1; SMN2ALDH1A1KMT2AUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3424928-A1 NITROGENOUS HETEROCYCLIC COMPOUND, PREPARATION METHOD, INTERMEDIATE, COMPOSITION AND USE Shanghai Pharmaceuticals Holding Co., Ltd. (CN) 2019-01-09 EP disclosed