SCHEMBL20644693

SCHEMBL20644693

Cc1cncc(C)c1N1CCC2(CC1)CNC(=O)O2

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CDK8 P49336 11/20 0.54
CDK19 Q9BWU1 11/20 0.54
CCNC P24863 7/20 0.53
SMO Q99835 1/20 0.49
LMNA P02545 1/20 0.44
CHRM2 P08172 1/20 0.44
ADRA2A P08913 1/20 0.44
CYP2D6 P10635 1/20 0.44
TSHR P16473 1/20 0.44
DRD1 P21728 1/20 0.44
CYP11B2 P19099 1/20 0.43
MAPT P10636 1/20 0.43
KMT2A Q03164 1/20 0.43
HDAC1 Q13547 1/20 0.41
EED O75530 1/20 0.38
PTPN11 Q06124 1/20 0.38
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
SLC6A3 Q01959 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18758215 0.91 CDK8 (0.50) CDK8CDK19CCNCSMOLMNA
SCHEMBL17113511 0.83 CDK8 (0.52) CDK8CDK19CCNCSMOLMNA
SCHEMBL18747990 0.78 CDK8 (0.59) CDK8CDK19CCNCSMOLMNA
SCHEMBL17129033 0.78 CDK8 (0.60) CDK8CDK19CCNCSMOLMNA
SCHEMBL17113642 0.75 CDK8 (0.62) CDK8CDK19CCNCSMOLMNA
SCHEMBL760272 0.74 LMNA (0.49) CDK8CDK19CCNCSMOLMNA
SCHEMBL1096010 0.72 LMNA (0.55) CDK8CDK19CCNCSMOLMNA
SCHEMBL17129049 0.72 CDK8 (1.00) CDK8CDK19CCNCHDAC1
SCHEMBL18747994 0.71 CDK8 (1.00) CDK8CDK19CCNC
SCHEMBL6683284 0.71 CYP2D6 (0.62) CDK8CDK19CCNCSMOLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3122739-B1 PYRIDYL PIPERIDINES MERCK PATENT GMBH (DE) 2019-01-16 EP disclosed