SCHEMBL20645796

SCHEMBL20645796

Cc1ccc(S(=O)(=O)N/N=C2\CCn3c2nc(C)c3Cl)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.46
HTR1A P08908 1/20 0.43
HTR2A P28223 1/20 0.43
HTR7 P34969 1/20 0.43
HTR6 P50406 1/20 0.43
KMT2A Q03164 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
MEN1 O00255 1/20 0.38
HTT P42858 1/20 0.38
F2 P00734 1/20 0.38
PRSS1 P07477 1/20 0.38
PRSS2 P07478 1/20 0.38
PRSS3 P35030 1/20 0.38
XBP1 P17861 1/20 0.38
EGFR P00533 1/20 0.37
KDM4E B2RXH2 1/20 0.37
MAPT P10636 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HIF1A Q16665 1/20 0.36
RECQL P46063 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20645794 0.88 ALDH1A1 (0.44) ALDH1A1HTR1AHTR2AHTR7HTR6
SCHEMBL20640753 0.88 ALDH1A1 (0.44) ALDH1A1HTR1AHTR2AHTR7HTR6
SCHEMBL8824083 0.71 PARP1 (0.48) ALDH1A1HTR1AHTR2AHTR7HTR6
SCHEMBL8824079 0.71 PARP1 (0.48) ALDH1A1HTR1AHTR2AHTR7HTR6
SCHEMBL31693805 0.67 ALDH1A1 (0.64) ALDH1A1KMT2AMEN1HTTF2
SCHEMBL30366023 0.66 ALDH1A1 (0.65) ALDH1A1HTR1AHTR2AHTR7HTR6
SCHEMBL19403826 0.66 ALDH1A1 (0.69) ALDH1A1HTR1AHTR2AHTR7HTR6
SCHEMBL20556203 0.65 ALDH1A1 (0.71) ALDH1A1KMT2AMEN1HTTF2
SCHEMBL16866377 0.65 ALDH1A1 (0.71) ALDH1A1KMT2AMEN1HTTF2
SCHEMBL17540297 0.64 ALDH1A1 (0.64) ALDH1A1KMT2ANPSR1MEN1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3652178-B1 BICYCLIC KETONE COMPOUNDS AND METHODS OF USE THEREOF HOFFMANN LA ROCHE (CH) 2024-01-24 EP disclosed
WO-2019012063-A1 BICYCLIC KETONE COMPOUNDS AND METHODS OF USE THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2019-01-17 WO disclosed