SCHEMBL2066098

SCHEMBL2066098

COc1ccc(CCN2CCC3CCCC=C3C2)cc1

nearest known ligand 0.55

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.55
SIGMAR1 Q99720 2/20 0.54
MAOA P21397 1/20 0.49
MAOB P27338 1/20 0.49
HTR1A P08908 1/20 0.46
SLC6A4 P31645 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acetic Acid SCHEMBL10926100 0.81 SIGMAR1 (0.47) HRH3SIGMAR1
SCHEMBL3219828 0.75 SIGMAR1 (0.47) HRH3SIGMAR1MAOAMAOBHTR1A
SCHEMBL12023880 0.73 SIGMAR1 (0.75) HRH3SIGMAR1HTR1ASLC6A4
SCHEMBL29356024 0.72 HRH3 (1.00) HRH3SIGMAR1MAOAMAOBSLC6A4
SCHEMBL10499190 0.72 SIGMAR1 (0.73) HRH3SIGMAR1MAOAMAOBHTR1A
SCHEMBL2066095 0.72 BCHE (0.44) HRH3SIGMAR1
SCHEMBL11156977 0.71 HRH3 (0.96) HRH3SIGMAR1MAOAMAOBSLC6A4
SCHEMBL9881343 0.70 SIGMAR1 (0.65) HRH3SIGMAR1MAOAMAOBHTR1A
SCHEMBL3590302 0.70 SIGMAR1 (0.69) HRH3SIGMAR1HTR1ASLC6A4
SCHEMBL6795798 0.70 SIGMAR1 (0.64) HRH3SIGMAR1MAOAMAOBHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2628728-B1 PROCESS FOR THE OPTICAL RESOLUTION OF 1-(4-METHOXYBENZYL)-OCTAHYDROISOQUINOLINE DIVI'S LABORATORIES LTD (IN) 2017-04-19 EP disclosed
CN-103319406-A Resolution of 1-(4-methoxybenzyl)-octahydro-isoquinoline DIVIS LAB LTD 2013-09-25 CN disclosed
EP-2628728-A1 Process for the optical resolution of 1-(4-methoxybenzyl)-octahydro-isoquinoline Divi's Laboratories Limited (IN) 2013-08-21 EP disclosed
US-8148527-B1 Resolution of 1-(4-methoxybenzyl)-octahydro-isoquinoline Divi's Laboratories, Ltd. (IN) 2012-04-03 US disclosed