SCHEMBL2066535

SCHEMBL2066535

O=C(O)Cc1cc(Cl)cc(Oc2ccc(S(=O)(=O)c3ccccc3)cc2Cl)c1

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 16/20 0.54
CHRM1 P11229 1/20 0.44
EPAS1 Q99814 1/20 0.44
PTGDR Q13258 1/20 0.44
FFAR1 O14842 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2065427 0.89 PTGDR2 (0.52) PTGDR2EPAS1PTGDR
SCHEMBL2066232 0.87 PTGDR2 (0.50) PTGDR2CHRM1EPAS1PTGDR
SCHEMBL883832 0.86 FFAR1 (0.46) PTGDR2EPAS1FFAR1
SCHEMBL2065895 0.86 PTGDR2 (0.50) PTGDR2EPAS1
SCHEMBL2066119 0.86 PTGDR2 (0.52) PTGDR2EPAS1
SCHEMBL586570 0.86 PTGDR2 (0.54) PTGDR2EPAS1PTGDRFFAR1
SCHEMBL2065952 0.85 PTGDR2 (0.55) PTGDR2EPAS1PTGDRFFAR1
SCHEMBL883850 0.82 PTGDR2 (0.48) PTGDR2EPAS1PTGDR
SCHEMBL883831 0.80 EPAS1 (0.47) PTGDR2EPAS1PTGDRFFAR1
SCHEMBL14490980 0.78 FFAR1 (0.42) PTGDR2EPAS1FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8148572-B2 Compounds ASTRAZENECA AB (SE) 2012-04-03 US claimed
US-20090192163-A1 Novel Compounds ASTRAZENECA AB (SE) 2009-07-30 US claimed
US-8148572-B2 Compounds ASTRAZENECA AB (SE) 2012-04-03 US disclosed
US-8148572-B2 Compounds ASTRAZENECA AB (SE) 2012-04-03 US disclosed
US-8148572-B2 Compounds ASTRAZENECA AB (SE) 2012-04-03 US disclosed
US-20090192163-A1 Novel Compounds ASTRAZENECA AB (SE) 2009-07-30 US disclosed
US-20090192163-A1 Novel Compounds ASTRAZENECA AB (SE) 2009-07-30 US disclosed
US-20090192163-A1 Novel Compounds ASTRAZENECA AB (SE) 2009-07-30 US disclosed
WO-2007039736-A1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2007-04-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090192163-A1 Novel Compounds PAH, PC, DDC PTGDR2 1000/4885CHRM1 1013/4885EPAS1 864/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.