SCHEMBL2069707

SCHEMBL2069707

Cc1cc(N(Cc2ccc(C(F)(F)F)cc2)C(=O)OC(C)(C)C)ccc1N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.41
PDK4 Q16654 1/20 0.41
PDK1 Q15118 1/20 0.38
HDAC6 Q9UBN7 3/20 0.38
HDAC1 Q13547 2/20 0.38
HDAC5 Q9UQL6 1/20 0.38
S100B P04271 1/20 0.38
LTB4R2 Q9NPC1 2/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.37
BCL2A1 Q16548 1/20 0.37
SERPINE1 P05121 2/20 0.36
LSS P48449 1/20 0.36
HDAC8 Q9BY41 1/20 0.35
STAT5B P51692 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
MAPK1 P28482 1/20 0.35
SIRT5 Q9NXA8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3609897 0.89 PDK2 (0.39) PDK2PDK4PDK1HDAC6HDAC1
SCHEMBL23609272 0.86 STAT5B (0.46) PDK2PDK4PDK1HDAC1S100B
SCHEMBL2070045 0.83 CYP19A1 (0.43) PDK2PDK4PDK1HDAC6HDAC1
SCHEMBL3604936 0.81 MMP1 (0.37) PDK2PDK4PDK1HDAC6HDAC1
SCHEMBL12252112 0.78 PDK2 (0.41) PDK2PDK4PDK1HDAC6BCL2A1
SCHEMBL24497425 0.78 ALDH1A1 (0.38) PDK2PDK4PDK1LTB4R2LSS
SCHEMBL29648358 0.77 LSS (0.35) PDK2PDK4PDK1HDAC6LTB4R2
SCHEMBL24497370 0.77 LSS (0.35) PDK2PDK4PDK1HDAC6LTB4R2
SCHEMBL23579129 0.76 STAT5B (0.43) HDAC1STAT5BMEN1KMT2AALDH1A1
SCHEMBL2072057 0.76 ALDH1A1 (0.46) MEN1KMT2AALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7906537-B2 Substituted p-diaminobenzene derivatives H. LUNDBECK A/S (DK) 2011-03-15 US disclosed
US-20060183791-A1 Substituted p-diaminobenzene derivatives H. LUNDBECK A/S (DK) 2006-08-17 US disclosed
EP-1613303-A1 SUBSTITUTED P-DIAMINOBENZENE DERIVATIVES H. Lundbeck A/S (DK) 2006-01-11 EP disclosed
WO-2004082677-A1 SUBSTITUTED P-DIAMINOBENZENE DERIVATIVES H. LUNDBECK A/S (DK) 2004-09-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060183791-A1 Substituted p-diaminobenzene derivatives ABCB1, UGT2B7, CYP2D6 PDK2 39/4885PDK4 171/4885PDK1 65/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.