SCHEMBL20711069

SCHEMBL20711069

CCCCN(C)C(=O)c1ccc2ccoc2c1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 2/20 0.47
HTR1B P28222 1/20 0.46
ALDH1A1 P00352 3/20 0.44
HPGD P15428 4/20 0.42
TSHR P16473 2/20 0.42
GAA P10253 2/20 0.42
CYP1A2 P05177 1/20 0.42
NAMPT P43490 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
KDM4E B2RXH2 2/20 0.38
LMNA P02545 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
PKM P14618 1/20 0.38
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL827802 0.79 HTR1B (0.55) PDK2HTR1BALDH1A1HPGDKDM4E
SCHEMBL9130521 0.77 PDK2 (0.54) PDK2ALDH1A1HPGDTSHRGAA
SCHEMBL23234372 0.76 MRGPRX4 (0.48) HTR1BALDH1A1HPGDTSHR
SCHEMBL25477867 0.74 HTR1B (0.50) HTR1BKDM4E
SCHEMBL30427249 0.74 CTNNB1 (0.56) HTR1BALDH1A1HPGDL3MBTL1NPC1
SCHEMBL827672 0.74 CTNNB1 (0.56) HTR1BALDH1A1HPGDL3MBTL1NPC1
SCHEMBL30427164 0.73 HTR1B (0.55) HTR1BALDH1A1L3MBTL1NPC1RAB9A
SCHEMBL14135299 0.73 HTR1B (0.55) HTR1BALDH1A1L3MBTL1NPC1RAB9A
SCHEMBL14233766 0.71 ALDH1A1 (0.52) PDK2ALDH1A1HPGDTSHRGAA
SCHEMBL24111798 0.71 HTR1B (0.64) HTR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019026014-A1 PROCESSES FOR PREPARATION OF LIFITEGRAST AND INTERMEDIATES THEREOF DR. REDDY'S LABORATORIES LIMITED (IN) 2019-02-07 WO disclosed