SCHEMBL20714701

SCHEMBL20714701

O=C(O)c1cc(Cl)cnc1Br

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.47
ALDH1A1 P00352 2/20 0.44
TP53 P04637 1/20 0.44
SORT1 Q99523 1/20 0.43
HCAR2 Q8TDS4 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
AKR1C4 P17516 1/20 0.42
AKR1C3 P42330 1/20 0.42
AKR1C2 P52895 1/20 0.42
AKR1C1 Q04828 1/20 0.42
DHODH Q02127 3/20 0.41
CYP3A4 P08684 1/20 0.41
DYRK1A Q13627 1/20 0.40
TSHR P16473 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
CASP1 P29466 1/20 0.39
GAA P10253 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18124622 0.82 KDR (0.49) KDRALDH1A1SORT1HCAR2TSHR
SCHEMBL3220148 0.82 KDR (0.46) KDRALDH1A1CASP1GAAPLAU
SCHEMBL1505655 0.79 KDM4E (0.45) ALDH1A1SORT1HCAR2AKR1C4AKR1C3
SCHEMBL915781 0.79 SMN1; SMN2 (0.48) ALDH1A1TP53SORT1HCAR2CA1
SCHEMBL29378297 0.79 SMN1; SMN2 (0.48) ALDH1A1TP53SORT1HCAR2CA1
SCHEMBL19682934 0.78 KDR (0.49) KDRALDH1A1LMNAKDM4E
SCHEMBL27836576 0.78 KDR (0.43) KDRALDH1A1CYP3A4SMN1; SMN2HPGD
SCHEMBL9684853 0.78 ALDH1A1 (0.45) ALDH1A1TP53SORT1HCAR2CA1
Hydrochloric Acid SCHEMBL6988496 0.78 SMN1; SMN2 (0.47) ALDH1A1TP53SORT1HCAR2CA1
SCHEMBL329752 0.78 CA1 (0.48) ALDH1A1TP53SORT1HCAR2CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118324761-A USP inhibitor, preparation method and application thereof 北京华森英诺生物科技有限公司 2024-07-12 CN disclosed
EP-3661928-B1 N-[(PYRIMIDINYLAMINO)PROPANYL]-, N-[(PYRIDYLAMINO)PROPANYL]- AND N-[(PYRAZINYLAMINO)PROPANYL]ARYLCARBOXAMIDES BOEHRINGER INGELHEIM INT (DE) 2021-06-16 EP disclosed
WO-2019025275-A1 NOVEL N-[(PYRIMIDINYLAMINO)PROPANYL]-, N-[(PYRIDYLAMINO)PROPANYL] - AND N-[(PYRAZINYLAMINO)PROPANYL]ARYLCARBOXAMIDES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2019-02-07 WO disclosed