SCHEMBL20718898

SCHEMBL20718898

C=Cc1nnnnc1NN

nearest known ligand 0.30

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.30
ADORA3 P0DMS8 1/20 0.30
MAPT P10636 1/20 0.30
MAOA P21397 1/20 0.30
PTGS1 P23219 1/20 0.30
OPRM1 P35372 1/20 0.30
KCNH2 Q12809 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31663430 0.73
SCHEMBL20718919 0.62
SCHEMBL21306180 0.60
SCHEMBL3622126 0.59
Fluoride SCHEMBL19062502 0.58
SCHEMBL5670604 0.53
SCHEMBL21306223 0.53
Bicarbonate SCHEMBL21633516 0.52 ALDH1A1 (0.30) ALDH1A1ADORA3MAPTMAOAPTGS1
SCHEMBL4623398 0.50
SCHEMBL873036 0.47 HDAC8 (0.32) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200182863-A1 NOVEL ANTIBODY CONJUGATES SUITABLE FOR USE IN DISCRETE FLUORESCENCE QUENCHING DISPLACEMENT IMMUNOASSAYS LIFE SCIENCE INKUBATOR SACHSEN GMBH & CO. KG (DE) 2020-06-11 US claimed
EP-3441766-B1 NOVEL ANTIBODY CONJUGATES SUITABLE FOR USE IN DISCRETE FLUORESCENCE QUENCHING DISPLACEMENT IMMUNOASSAYS LIFE SCIENCE INKUBATOR SACHSEN GMBH & CO KG (DE) 2020-03-11 EP claimed
EP-3441766-A1 NOVEL ANTIBODY CONJUGATES SUITABLE FOR USE IN DISCRETE FLUORESCENCE QUENCHING DISPLACEMENT IMMUNOASSAYS Life Science Inkubator Sachsen GmbH & Co. KG (DE) 2019-02-13 EP claimed
US-20200182863-A1 NOVEL ANTIBODY CONJUGATES SUITABLE FOR USE IN DISCRETE FLUORESCENCE QUENCHING DISPLACEMENT IMMUNOASSAYS LIFE SCIENCE INKUBATOR SACHSEN GMBH & CO. KG (DE) 2020-06-11 US disclosed
EP-3441766-B1 NOVEL ANTIBODY CONJUGATES SUITABLE FOR USE IN DISCRETE FLUORESCENCE QUENCHING DISPLACEMENT IMMUNOASSAYS LIFE SCIENCE INKUBATOR SACHSEN GMBH & CO KG (DE) 2020-03-11 EP disclosed
WO-2019030287-A1 NOVEL ANTIBODY CONJUGATES SUITABLE FOR USE IN DISCRETE FLUORESCENCE QUENCHING DISPLACEMENT IMMUNOASSAYS LIFE SCIENCE INKUBATOR SACHSEN GMBH & CO. KG (DE) 2019-02-14 WO disclosed
EP-3441766-A1 NOVEL ANTIBODY CONJUGATES SUITABLE FOR USE IN DISCRETE FLUORESCENCE QUENCHING DISPLACEMENT IMMUNOASSAYS Life Science Inkubator Sachsen GmbH & Co. KG (DE) 2019-02-13 EP disclosed