SCHEMBL2071971

SCHEMBL2071971

COC(=O)CSc1cccc(F)c1C#N

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.59
MAPT P10636 7/20 0.59
HPGD P15428 7/20 0.59
HSD17B10 Q99714 6/20 0.59
TP53 P04637 2/20 0.59
KDM4E B2RXH2 6/20 0.52
CYP2C19 P33261 3/20 0.52
CYP1A2 P05177 2/20 0.52
CYP3A4 P08684 2/20 0.52
CYP2C9 P11712 2/20 0.52
GLA P06280 1/20 0.52
GAA P10253 1/20 0.52
L3MBTL1 Q9Y468 3/20 0.50
POLB P06746 2/20 0.50
PKM P14618 1/20 0.46
TSHR P16473 3/20 0.45
MAPK1 P28482 2/20 0.45
RAB9A P51151 3/20 0.43
NPC1 O15118 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8238275 0.81 ALDH1A1 (0.57) ALDH1A1MAPTHPGDHSD17B10TP53
SCHEMBL26968212 0.78 HSD17B10 (0.54) ALDH1A1MAPTHPGDHSD17B10TP53
SCHEMBL4420424 0.75 MAPT (0.56) ALDH1A1MAPTHPGDHSD17B10TP53
SCHEMBL8153543 0.74 HSD17B10 (0.63) ALDH1A1MAPTHPGDHSD17B10TP53
SCHEMBL18496514 0.73 ALDH1A1 (0.48) ALDH1A1MAPTHPGDHSD17B10TP53
SCHEMBL25575139 0.72 MAPT (0.75) ALDH1A1MAPTHPGDHSD17B10TP53
SCHEMBL3338630 0.71 HSD17B10 (0.46) ALDH1A1MAPTHPGDHSD17B10TP53
SCHEMBL846222 0.70 ALDH1A1 (0.41) ALDH1A1HPGDHSD17B10KDM4EL3MBTL1
SCHEMBL8144828 0.69 HSD17B10 (0.66) ALDH1A1MAPTHPGDHSD17B10TP53
SCHEMBL11544945 0.68 HSD17B10 (0.64) ALDH1A1MAPTHPGDHSD17B10TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7863444-B2 4-aminopyrrolopyrimidines as kinase inhibitors ABBOTT LABORATORIES (US) 2011-01-04 US disclosed