SCHEMBL20740673

SCHEMBL20740673

COC(=O)c1ccc(OCCCOc2c(C)nc(N)nc2N)cc1

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DHFR P00374 7/20 0.60
MAPT P10636 5/20 0.56
RAB9A P51151 2/20 0.51
SLC2A1 P11166 1/20 0.49
TDP1 Q9NUW8 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
GLA P06280 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
NPC1 O15118 1/20 0.46
TP53 P04637 1/20 0.46
MAPK1 P28482 1/20 0.46
KMT2A Q03164 3/20 0.44
TSHR P16473 1/20 0.44
ALDH1A1 P00352 2/20 0.44
KDM4E B2RXH2 1/20 0.44
LMNA P02545 1/20 0.44
HPGD P15428 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20740677 0.87 DHFR (0.69) DHFRSLC2A1TP53TSHR
SCHEMBL20740676 0.86 DHFR (0.48) DHFRSLC2A1TP53MAPK1TSHR
SCHEMBL2469151 0.79 MAPT (0.89) MAPTRAB9ATDP1L3MBTL1SMN1; SMN2
SCHEMBL20740672 0.78 DHFR (0.56) DHFRMAPTSLC2A1SMN1; SMN2KMT2A
SCHEMBL20740670 0.78 DHFR (0.53) DHFRRAB9ASLC2A1SMN1; SMN2NPC1
SCHEMBL11171761 0.77 DHFR (0.57) DHFRMAPTSLC2A1KMT2AALDH1A1
SCHEMBL11171619 0.77 DHFR (0.57) DHFRMAPTSLC2A1KMT2AALDH1A1
Hydrochloric Acid SCHEMBL11185095 0.76 DHFR (0.56) DHFRMAPTSLC2A1KMT2AALDH1A1
SCHEMBL20740675 0.76 KMT2A (0.54) DHFRSLC2A1KMT2A
SCHEMBL1796892 0.75 MAPT (0.79) MAPTRAB9ATDP1L3MBTL1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2194985-B1 ANTIMALARIAL COMPOUNDS WITH FLEXIBLE SIDE-CHAINS MEDICINES FOR MALARIA VENTURE MMV (CH) 2019-02-20 EP claimed
EP-2194985-B1 ANTIMALARIAL COMPOUNDS WITH FLEXIBLE SIDE-CHAINS MEDICINES FOR MALARIA VENTURE MMV (CH) 2019-02-20 EP disclosed