SCHEMBL20740677

SCHEMBL20740677

Cc1nc(N)nc(N)c1OCCCOc1ccc(C(=O)O)cc1

nearest known ligand 0.69

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DHFR P00374 8/20 0.69
PLA2G4B P0C869 2/20 0.52
TP53 P04637 1/20 0.50
TSHR P16473 1/20 0.50
SLC2A1 P11166 1/20 0.48
PKM P14618 1/20 0.48
RARB P10826 3/20 0.47
HTT P42858 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20740673 0.87 DHFR (0.60) DHFRTP53TSHRSLC2A1
SCHEMBL31155811 0.86 DHFR (0.91) DHFRPLA2G4BTP53TSHRHTT
SCHEMBL20740675 0.85 KMT2A (0.54) DHFRPLA2G4BSLC2A1
SCHEMBL20740670 0.85 DHFR (0.53) DHFRSLC2A1
SCHEMBL20740678 0.80 DHFR (0.52) DHFRSLC2A1
SCHEMBL11171761 0.79 DHFR (0.57) DHFRSLC2A1
Hydrochloric Acid SCHEMBL11185095 0.78 DHFR (0.56) DHFRSLC2A1
SCHEMBL20740668 0.77 DHFR (0.58) DHFRSLC2A1HTT
SCHEMBL118037 0.76 PKM (0.77) PLA2G4BTP53TSHRPKMRARB
SCHEMBL20740676 0.76 DHFR (0.48) DHFRTP53TSHRSLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2194985-B1 ANTIMALARIAL COMPOUNDS WITH FLEXIBLE SIDE-CHAINS MEDICINES FOR MALARIA VENTURE MMV (CH) 2019-02-20 EP claimed
EP-2194985-B1 ANTIMALARIAL COMPOUNDS WITH FLEXIBLE SIDE-CHAINS MEDICINES FOR MALARIA VENTURE MMV (CH) 2019-02-20 EP disclosed