SCHEMBL2074903

SCHEMBL2074903

CC(C)N1CCN(c2cc(NC(=O)N3Cc4ccccc4C3)ncn2)CC1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.49
KCNH2 Q12809 1/20 0.49
SCN9A Q15858 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.47
NAMPT P43490 9/20 0.47
NPC1 O15118 1/20 0.46
ALDH1A1 P00352 1/20 0.46
ATM Q13315 1/20 0.46
HRH4 Q9H3N8 1/20 0.45
LOXL2 Q9Y4K0 1/20 0.44
TAS1R3 Q7RTX0 1/20 0.43
TAS1R1 Q7RTX1 1/20 0.43
TAS1R2 Q8TE23 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2073745 0.85 SMN1; SMN2 (0.49) SMN1; SMN2NPC1ALDH1A1ATMLOXL2
SCHEMBL2074775 0.85 HDAC3 (0.50) SCN9ASMN1; SMN2NAMPTNPC1ALDH1A1
SCHEMBL2074790 0.84 SMN1; SMN2 (0.51) SMN1; SMN2NPC1ALDH1A1ATMLOXL2
SCHEMBL2075861 0.84 SMN1; SMN2 (0.51) SMN1; SMN2NPC1ALDH1A1ATMLOXL2
SCHEMBL2075728 0.83 SMN1; SMN2 (0.52) SCN9ASMN1; SMN2NPC1ALDH1A1ATM
SCHEMBL2074244 0.82 NPC1 (0.53) SMN1; SMN2NPC1ALDH1A1ATM
SCHEMBL2075431 0.81 LMNA (0.43) HRH3SMN1; SMN2NPC1ALDH1A1ATM
SCHEMBL2075521 0.81 NAMPT (0.53) HRH3KCNH2SCN9ASMN1; SMN2NAMPT
SCHEMBL2075500 0.78 SMN1; SMN2 (0.42) HRH3SMN1; SMN2ALDH1A1
SCHEMBL2072344 0.77 CNR2 (0.43) HRH3SMN1; SMN2ALDH1A1LOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7902184-B2 Piperazinyl pyrimidine derivatives HOFFMANN-LA ROCHE INC. (US) 2011-03-08 US disclosed