SCHEMBL20749376

SCHEMBL20749376

CCCSN(c1cc(F)c(F)c(C(=O)c2ccc3ncc(N4CCOCC4)nc3c2)c1F)S(=O)(=O)CCC

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CDK6 Q00534 2/20 0.37
HPGD P15428 1/20 0.36
PIK3CD O00329 11/20 0.36
PIK3CA P42336 11/20 0.36
PIK3CB P42338 11/20 0.36
PIK3CG P48736 10/20 0.36
MTOR P42345 6/20 0.36
PRKDC P78527 1/20 0.36
PIK3C3 Q8NEB9 1/20 0.36
BRAF P15056 1/20 0.36
FGFR2 P21802 1/20 0.34
FGFR3 P22607 1/20 0.34
SHMT2 P34897 2/20 0.33
NPC1 O15118 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14715976 0.89 CDK6 (0.39) CDK6HPGDPIK3CDPIK3CAPIK3CB
SCHEMBL29623943 0.89 CDK6 (0.39) CDK6HPGDPIK3CDPIK3CAPIK3CB
SCHEMBL20749375 0.84 BRAF (0.30) BRAF
SCHEMBL20749382 0.83 CDK6 (0.37) CDK6HPGDPIK3CDPIK3CAPIK3CB
SCHEMBL20749349 0.80 HPGD (0.40) HPGDBRAFNPC1
Uplarafenib SCHEMBL14716189 0.80 BRAF (0.51) CDK6HPGDPIK3CDPIK3CAPIK3CB
Uplarafenib SCHEMBL29623930 0.80 BRAF (0.51) CDK6HPGDPIK3CDPIK3CAPIK3CB
SCHEMBL20749378 0.79 CDK6 (0.41) CDK6HPGDPIK3CDPIK3CAPIK3CB
SCHEMBL29624095 0.78 HPGD (0.42) CDK6HPGDPIK3CDPIK3CAPIK3CB
SCHEMBL14829458 0.77 HPGD (0.46) CDK6HPGDPIK3CDPIK3CAPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2747767-B1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS NEUPHARMA INC (US) 2019-02-20 EP disclosed