SCHEMBL20765247

SCHEMBL20765247

O=C1CCC(N2Cc3cc(C4CCN(Cc5ccccc5)CC4)ccc3C2=O)C(=O)N1

nearest known ligand 0.78

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
IKZF1 Q13422 6/20 0.78
IKZF2 Q9UKS7 14/20 0.77

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30368853 0.96 IKZF1 (0.73) IKZF1IKZF2
SCHEMBL20936143 0.96 IKZF1 (0.73) IKZF1IKZF2
SCHEMBL20765392 0.96 IKZF1 (0.73) IKZF1IKZF2
SCHEMBL20765806 0.96 IKZF1 (0.73) IKZF1IKZF2
SCHEMBL20765608 0.96 IKZF1 (0.73) IKZF1IKZF2
SCHEMBL23895451 0.96 IKZF1 (0.73) IKZF1IKZF2
SCHEMBL20765393 0.96 IKZF1 (0.73) IKZF1IKZF2
SCHEMBL20765811 0.96 IKZF1 (0.73) IKZF1IKZF2
SCHEMBL20765691 0.96 IKZF1 (0.73) IKZF1IKZF2
SCHEMBL30368942 0.96 IKZF1 (0.73) IKZF1IKZF2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 51 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240335452-A1 COMPOSITIONS AND METHODS OF COMBINATION THERAPY FOR TARGETING LYMPHOMA CULLGEN (SHANGHAI), INC. (CN) 2024-10-10 US claimed
CN-118201612-A Compositions and methods for combination therapy for the treatment of lymphomas 上海睿跃生物科技有限公司 2024-06-14 CN claimed
CN-111051298-B 3- (1-oxo-isoindolin-2-yl) piperidine-2, 6-dione derivative and application thereof 诺华股份有限公司 2023-06-27 CN claimed
EP-3672949-B9 3-(1-OXOISOINDOLIN-2-YL)PIPERIDINE-2,6-DIONE DERIVATIVES AND USES THEREOF NOVARTIS AG (CH) 2023-04-05 EP claimed
EP-3672949-B1 3-(1-OXOISOINDOLIN-2-YL)PIPERIDINE-2,6-DIONE DERIVATIVES AND USES THEREOF NOVARTIS AG (CH) 2022-12-21 EP claimed
US-20210309638-A1 3-(1-OXOISOINDOLIN-2-YL)PIPERIDINE-2,6-DIONE DERIVATIVES AND USES THEREOF NOVARTIS AG (CH) 2021-10-07 US claimed
US-20200231569-A1 3-(1-OXOISOINDOLIN-2-YL)PIPERIDINE-2,6-DIONE DERIVATIVES AND USES THEREOF NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, INC. 2020-07-23 US claimed
EP-3672949-A1 3-(1-OXOISOINDOLIN-2-YL)PIPERIDINE-2,6-DIONE DERIVATIVES AND USES THEREOF Novartis AG (CH) 2020-07-01 EP claimed
CN-111051298-A 3- (1-oxoisoindolin-2-yl) piperidine-2, 6-dione derivatives and uses thereof 诺华股份有限公司 2020-04-21 CN claimed
US-10414755-B2 3-(1-oxoisoindolin-2-yl)piperidine-2,6-dione derivatives and uses thereof NOVARTIS AG (CH) 2019-09-17 US claimed
WO-2019038717-A1 3-(1-OXOISOINDOLIN-2-YL)PIPERIDINE-2,6-DIONE DERIVATIVES AND USES THEREOF NOVARTIS AG (CH) 2019-02-28 WO claimed
US-20240384007-A1 COMPOSITIONS AND METHODS FOR SELECTIVE PROTEIN DEGRADATION NOVARTIS AG (CH) 2024-11-21 US disclosed
US-20240376096-A1 SMALL MOLECULE CYCLIN DEPENDENT KINASE 4/6 (CDK4/6) AND IKZF2 (HELIOS) DEGRADERS AND METHODS OF USE THEREOF DANA-FARBER CANCER INSTITUTE, INC. (US) 2024-11-14 US disclosed
US-20240335452-A1 COMPOSITIONS AND METHODS OF COMBINATION THERAPY FOR TARGETING LYMPHOMA CULLGEN (SHANGHAI), INC. (CN) 2024-10-10 US disclosed
CN-118201612-A Compositions and methods for combination therapy for the treatment of lymphomas 上海睿跃生物科技有限公司 2024-06-14 CN disclosed
US-10640489-B2 3-(1-oxoisoindolin-2-yl)piperidine-2,6-dione derivatives and uses thereof NOVARTIS AG (CH) 2020-05-05 US disclosed
CN-111051298-A 3- (1-oxoisoindolin-2-yl) piperidine-2, 6-dione derivatives and uses thereof 诺华股份有限公司 2020-04-21 CN disclosed
US-10414755-B2 3-(1-oxoisoindolin-2-yl)piperidine-2,6-dione derivatives and uses thereof NOVARTIS AG (CH) 2019-09-17 US disclosed
US-10414755-B2 3-(1-oxoisoindolin-2-yl)piperidine-2,6-dione derivatives and uses thereof NOVARTIS AG (CH) 2019-09-17 US disclosed
WO-2019079569-A1 COMPOSITIONS AND METHODS FOR SELECTIVE PROTEIN DEGRADATION NOVARTIS AG (CH) 2019-04-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10414755-B2 3-(1-oxoisoindolin-2-yl)piperidine-2,6-dione derivatives and uses thereof XDH, H1-0, RXFP1 IKZF1 3202/4885IKZF2 4353/4885
US-20240376096-A1 SMALL MOLECULE CYCLIN DEPENDENT KINASE 4/6 (CDK4/6) AND IKZF2 (HELIOS) DEGRADERS AND METHODS OF USE THEREOF IKZF2, CDK6, IKZF1 IKZF1 3/4885IKZF2 1/4885
US-20240384007-A1 COMPOSITIONS AND METHODS FOR SELECTIVE PROTEIN DEGRADATION CRBN, RPS27A, COPB1 IKZF1 781/4885IKZF2 336/4885
US-10640489-B2 3-(1-oxoisoindolin-2-yl)piperidine-2,6-dione derivatives and uses thereof XDH, H1-0, RXFP1 IKZF1 3202/4885IKZF2 4353/4885
US-20210309638-A1 3-(1-OXOISOINDOLIN-2-YL)PIPERIDINE-2,6-DIONE DERIVATIVES AND USES THEREOF XDH, H1-0, RXFP1 IKZF1 3202/4885IKZF2 4353/4885
US-20240335452-A1 COMPOSITIONS AND METHODS OF COMBINATION THERAPY FOR TARGETING LYMPHOMA EZH2, BCL6, BMI1 IKZF1 12/4885IKZF2 7/4885
US-20200231569-A1 3-(1-OXOISOINDOLIN-2-YL)PIPERIDINE-2,6-DIONE DERIVATIVES AND USES THEREOF XDH, H1-0, RXFP1 IKZF1 3202/4885IKZF2 4353/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.