SCHEMBL20765458

SCHEMBL20765458

Cc1nc2cc(C(=O)N3CCN(CCc4ccccc4)C[C@@H]3C(C)C)ccc2[nH]1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 2/20 0.42
ACHE P22303 2/20 0.42
HRH4 Q9H3N8 1/20 0.40
AGTR2 P50052 1/20 0.40
HSD11B1 P28845 2/20 0.39
RAB9A P51151 3/20 0.39
PARP1 P09874 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
KCNH2 Q12809 1/20 0.38
TLR9 Q9NR96 1/20 0.37
TLR8 Q9NR97 1/20 0.37
TLR7 Q9NYK1 1/20 0.37
TSSK1B Q9BXA7 1/20 0.36
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MAPK14 Q16539 1/20 0.36
NPC1 O15118 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20765461 1.00 BCHE (0.42) BCHEACHEHRH4AGTR2HSD11B1
SCHEMBL20765524 0.88 MAPK14 (0.44) BCHEACHEHRH4AGTR2HSD11B1
SCHEMBL20765527 0.88 MAPK14 (0.44) BCHEACHEHRH4AGTR2HSD11B1
SCHEMBL20765824 0.84 BCHE (0.41) BCHEACHEHSD11B1ALDH1A1POLB
SCHEMBL20765826 0.84 BCHE (0.41) BCHEACHEHSD11B1ALDH1A1POLB
SCHEMBL20765553 0.81 BRS3 (0.40) BCHEACHESMN1; SMN2MAPK14
SCHEMBL20765550 0.81 BRS3 (0.40) BCHEACHESMN1; SMN2MAPK14
SCHEMBL20765611 0.79 HSD11B1 (0.41) HSD11B1RAB9AMEN1KMT2AALDH1A1
SCHEMBL20765609 0.79 HSD11B1 (0.41) HSD11B1RAB9AMEN1KMT2AALDH1A1
SCHEMBL20766168 0.75 HPGD (0.43) BCHEACHERAB9AKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019038683-A1 COMPOUNDS TARGETING TANDEM BRCT DOMAINS OF BRCA1, COMPOSITIONS AND METHODS THEREOF INSTITUTE FOR STEM CELL BIOLOGY AND REGENERATIVE MEDICINE (IN) 2019-02-28 WO claimed