SCHEMBL20765482

SCHEMBL20765482

O=C(c1ccc2nc(-c3ccccc3)[nH]c2c1)N1CCN(C(=O)O)C(Cc2ccccc2)C1

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 1/20 0.56
BCHE P06276 2/20 0.51
ACHE P22303 2/20 0.51
CHEK2 O96017 6/20 0.49
CA1 P00915 10/20 0.48
CA2 P00918 10/20 0.48
CA4 P22748 10/20 0.48
CA9 Q16790 10/20 0.48
HPGD P15428 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19970784 0.77 MGLL (0.59) MGLLBCHEACHECHEK2HPGD
SCHEMBL21843704 0.77 HPGD (0.70) MGLLCHEK2HPGD
SCHEMBL16619560 0.76 MGLL (0.65) MGLLCHEK2HPGD
SCHEMBL19986744 0.75 MGLL (0.57) MGLLBCHEACHECHEK2HPGD
SCHEMBL16631031 0.73 MGLL (0.60) MGLLBCHEACHECHEK2HPGD
SCHEMBL20765523 0.72 MGLL (0.58) MGLLBCHEACHECHEK2HPGD
SCHEMBL20765507 0.72 CHEK2 (0.58) MGLLBCHEACHECHEK2HPGD
SCHEMBL20765786 0.72 BCHE (0.55) MGLLBCHEACHECHEK2
SCHEMBL19970751 0.72 BCHE (0.55) MGLLBCHEACHECHEK2
SCHEMBL20765497 0.72 MGLL (0.58) MGLLBCHEACHECHEK2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019038683-A1 COMPOUNDS TARGETING TANDEM BRCT DOMAINS OF BRCA1, COMPOSITIONS AND METHODS THEREOF INSTITUTE FOR STEM CELL BIOLOGY AND REGENERATIVE MEDICINE (IN) 2019-02-28 WO disclosed