SCHEMBL19986744

SCHEMBL19986744

O=C(c1ccc2nc(-c3ccccc3)[nH]c2c1)N1CCN(C(O)OCc2ccccc2)CC1

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 1/20 0.57
CHEK2 O96017 10/20 0.52
BCHE P06276 2/20 0.49
ACHE P22303 2/20 0.49
ACACB O00763 2/20 0.49
ACACA Q13085 1/20 0.47
PDE4A P27815 1/20 0.47
PDE4B Q07343 1/20 0.47
PDE4C Q08493 1/20 0.47
PDE4D Q08499 1/20 0.47
HPGD P15428 1/20 0.47
HDAC3 O15379 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19986737 0.92 ACACB (0.51) MGLLCHEK2BCHEACHEACACB
SCHEMBL19986696 0.88 ACACB (0.51) MGLLCHEK2ACACBHPGD
SCHEMBL19970784 0.85 MGLL (0.59) MGLLCHEK2BCHEACHEACACB
SCHEMBL21843704 0.79 HPGD (0.70) MGLLCHEK2ACACBACACAHPGD
SCHEMBL16619560 0.78 MGLL (0.65) MGLLCHEK2ACACBACACAHPGD
SCHEMBL19970809 0.78 ACACB (0.52) MGLLCHEK2BCHEACHEACACB
SCHEMBL19970783 0.78 ENPP2 (0.56) MGLLCHEK2ACACBHPGD
SCHEMBL20765523 0.75 MGLL (0.58) MGLLCHEK2BCHEACHEACACB
SCHEMBL20765482 0.75 MGLL (0.56) MGLLCHEK2BCHEACHEHPGD
SCHEMBL20765786 0.75 BCHE (0.55) MGLLCHEK2BCHEACHEACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3296297-A1 BENZIMIDAZOL DERIVATIVES FOR TREATING FILOVIRUS INFECTION CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2018-03-21 EP disclosed