SCHEMBL20765610

SCHEMBL20765610

O=C(OCc1ccccc1)N1CCN(Cc2ccc3cc[nH]c3c2)CC1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 3/20 0.65
MAPK14 Q16539 4/20 0.62
TSHR P16473 1/20 0.50
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
SMN1; SMN2 Q16637 2/20 0.47
NPC1 O15118 2/20 0.47
RAB9A P51151 1/20 0.47
FNTA P49354 2/20 0.46
FNTB P49356 2/20 0.46
PGGT1B P53609 2/20 0.46
ENPP2 Q13822 2/20 0.46
CYP2C19 P33261 1/20 0.46
TNKS O95271 1/20 0.45
PARP1 P09874 1/20 0.45
TNKS2 Q9H2K2 1/20 0.45
PARP2 Q9UGN5 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13150118 0.85 KMT2A (0.63) FAAHMEN1KMT2ANPSR1SMN1; SMN2
SCHEMBL20765500 0.83 MAPK14 (0.70) MAPK14TSHRMEN1KMT2ANPSR1
SCHEMBL3752475 0.82 FAAH (0.70) FAAHMAPK14TSHRNPC1ENPP2
SCHEMBL18935537 0.80 FAAH (0.58) FAAHMAPK14TSHR
SCHEMBL19970835 0.79 BCHE (0.53) TNKSPARP1TNKS2PARP2GRIN2B
SCHEMBL29132085 0.79 SIGMAR1 (0.59) FAAHMEN1KMT2ANPSR1SMN1; SMN2
SCHEMBL3597986 0.79 FAAH (1.00) FAAH
SCHEMBL23301159 0.78 KDM4E (0.65) FAAHTSHRMEN1KMT2ANPSR1
SCHEMBL29943050 0.78 KDM4E (0.65) FAAHTSHRMEN1KMT2ANPSR1
SCHEMBL20782366 0.78 MAPK14 (0.71) MAPK14MEN1KMT2ANPSR1ENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019038683-A1 COMPOUNDS TARGETING TANDEM BRCT DOMAINS OF BRCA1, COMPOSITIONS AND METHODS THEREOF INSTITUTE FOR STEM CELL BIOLOGY AND REGENERATIVE MEDICINE (IN) 2019-02-28 WO claimed