SCHEMBL20770802

SCHEMBL20770802

NC(=O)c1cccc(-c2ccccn2)c1-c1ncc[nH]1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK1A1 P48729 1/20 0.66
TYRO3 Q06418 1/20 0.66
DYRK1B Q9Y463 1/20 0.66
PARP1 P09874 4/20 0.47
GRM5 P41594 2/20 0.47
DHODH Q02127 1/20 0.46
PARP2 Q9UGN5 1/20 0.46
NUDT1 P36639 1/20 0.43
KEAP1 Q14145 1/20 0.42
NFE2L2 Q16236 1/20 0.42
BTK Q06187 1/20 0.40
AURKA O14965 1/20 0.40
BCAT2 O15382 1/20 0.40
ADRA1A P35348 1/20 0.39
KMT2A Q03164 1/20 0.39
TGFBR1 P36897 1/20 0.39
CDC7 O00311 1/20 0.39
CHEK2 O96017 1/20 0.38
MTOR P42345 1/20 0.37
ADK P55263 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL986588 0.82 CSNK1A1 (0.46) CSNK1A1TYRO3DYRK1BPARP1GRM5
SCHEMBL6825869 0.80 CSNK1A1 (1.00) CSNK1A1TYRO3DYRK1BPARP1GRM5
SCHEMBL2943452 0.80 GRM5 (0.54) CSNK1A1TYRO3DYRK1BPARP1GRM5
SCHEMBL4564863 0.79 CSNK1A1 (0.61) CSNK1A1TYRO3DYRK1BPARP1NUDT1
Water SCHEMBL30473073 0.79 CSNK1A1 (0.97) CSNK1A1TYRO3DYRK1BPARP1GRM5
SCHEMBL997865 0.78 GRM5 (0.64) CSNK1A1TYRO3DYRK1BPARP1GRM5
SCHEMBL29506339 0.78 GRM5 (0.64) CSNK1A1TYRO3DYRK1BPARP1GRM5
SCHEMBL31249988 0.78 GRM5 (0.64) CSNK1A1TYRO3DYRK1BPARP1GRM5
SCHEMBL31249984 0.78 GRM5 (0.64) CSNK1A1TYRO3DYRK1BPARP1GRM5
SCHEMBL986590 0.78 CSNK1A1 (0.47) CSNK1A1TYRO3DYRK1BPARP1GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019046303-A1 A METHOD FOR PREDICTING A SUBJECT'S RESPONSE TO SLC MODULATOR THERAPY THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2019-03-07 WO disclosed