SCHEMBL20780744

SCHEMBL20780744

NC(=O)/C=C/[C@H]1CCCN1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 2/20 0.36
NOS3 P29474 1/20 0.36
NOS1 P29475 1/20 0.36
KMT2A Q03164 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MAPT P10636 1/20 0.34
ATM Q13315 1/20 0.34
CYP2D6 P10635 1/20 0.34
GLI1 P08151 1/20 0.34
MEN1 O00255 1/20 0.34
BLM P54132 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29907711 1.00 NOS2 (0.36) NOS2NOS3NOS1KMT2AKDM4E
SCHEMBL29907713 1.00 NOS2 (0.36) NOS2NOS3NOS1KMT2AKDM4E
SCHEMBL29907813 1.00 NOS2 (0.36) NOS2NOS3NOS1KMT2AKDM4E
SCHEMBL26088434 0.82 MEN1 (0.40) KMT2AMAPTMEN1BLM
SCHEMBL22368106 0.82 MEN1 (0.40) KMT2AMAPTMEN1BLM
SCHEMBL26088431 0.82 MEN1 (0.40) KMT2AMAPTMEN1BLM
SCHEMBL21794634 0.80 SLC6A2 (0.35) KMT2AMEN1BLM
SCHEMBL18991730 0.79
SCHEMBL6819028 0.79
SCHEMBL20327088 0.77 SLC6A3 (0.33) KMT2AMAPTMEN1BLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3677583-A1 NITROGENOUS HETEROCYCLIC COMPOUND, PREPARATION METHOD, INTERMEDIATE, COMPOSITION, AND APPLICATION Shanghai Pharmaceuticals Holding Co., Ltd. (CN) 2020-07-08 EP disclosed
WO-2019042409-A1 NITROGENOUS HETEROCYCLIC COMPOUND, PREPARATION METHOD, INTERMEDIATE, COMPOSITION, AND APPLICATION 上海医药集团股份有限公司 2019-03-07 WO disclosed