SCHEMBL20780902

SCHEMBL20780902

C=C(O)c1nc(Cl)sc1-c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 4/20 0.40
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 2/20 0.39
HPGD P15428 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HSD17B10 Q99714 1/20 0.39
HCRTR1 O43613 1/20 0.38
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
MAPT P10636 1/20 0.37
CYP2C19 P33261 1/20 0.37
NPSR1 Q6W5P4 1/20 0.35
TDO2 P48775 1/20 0.34
GAA P10253 1/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20780956 0.82 ALDH1A1 (0.47) ALOX5ALDH1A1KDM4EHPGDSMN1; SMN2
SCHEMBL3315030 0.82 KDM4E (0.50) ALOX5ALDH1A1KDM4EHPGDSMN1; SMN2
SCHEMBL9587190 0.76 KDM4E (0.69) ALDH1A1KDM4EHPGDSMN1; SMN2HSD17B10
SCHEMBL13616800 0.76 ALDH1A1 (0.48) ALOX5ALDH1A1KDM4EHPGDSMN1; SMN2
SCHEMBL20780903 0.75 ALDH1A1 (0.47) ALOX5ALDH1A1KDM4EHPGDSMN1; SMN2
SCHEMBL11753179 0.73 ALDH1A1 (0.60) ALDH1A1KDM4EHPGDSMN1; SMN2CYP1A2
SCHEMBL3321548 0.72 GRM6 (0.58) ALDH1A1KDM4EHPGDSMN1; SMN2HSD17B10
SCHEMBL2186972 0.72 HPGD (0.51) ALDH1A1KDM4EHPGDSMN1; SMN2HSD17B10
SCHEMBL6800972 0.72 ALDH1A1 (0.54) ALOX5ALDH1A1KDM4EHPGDSMN1; SMN2
SCHEMBL9586464 0.71 HDAC3 (0.44) ALDH1A1KDM4EHPGDSMN1; SMN2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019043407-A1 SUBSTITUTED 2-AZABICYCLO[3.1.1]HEPTANE AND 2-AZABICYCLO[3.2.1]OCTANE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS CHRONOS THERAPEUTICS LIMITED (GB) 2019-03-07 WO disclosed