SCHEMBL20782875

SCHEMBL20782875

Cc1ccc2scc(N3CCN(C)CC3)c(=O)c2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAPT P10636 19/20 1.00
THRB P10828 2/20 1.00
USP2 O75604 2/20 1.00
TP53 P04637 10/20 0.78
LMNA P02545 2/20 0.74
POLB P06746 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22860672 0.88 MAPT (0.79) MAPTTHRBUSP2TP53LMNA
SCHEMBL9618122 0.77 MAPT (0.63) MAPTTHRBUSP2TP53LMNA
SCHEMBL23010594 0.72 MAPT (0.58) MAPTTHRBUSP2TP53LMNA
SCHEMBL8919052 0.72 MAPT (0.58) MAPTTHRBUSP2TP53LMNA
SCHEMBL4539425 0.70 MAPT (0.54) MAPTTHRBUSP2TP53LMNA
SCHEMBL10890683 0.69 MAPT (0.54) MAPTTHRBUSP2TP53LMNA
SCHEMBL22860673 0.69 MAPT (0.52) MAPTTHRBUSP2TP53LMNA
SCHEMBL20784531 0.67 MAPT (0.53) MAPTTHRBUSP2POLB
SCHEMBL13292998 0.67 MEN1 (0.57) MAPTTHRBUSP2TP53LMNA
SCHEMBL7923952 0.67 HTR1A (0.58) MAPTTHRBUSP2LMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10220016-B2 Methods and materials for assessing chemotherapy responsiveness and treating cancer MAYO FOUNDATION FOR MEDICAL EDUCATION AND RESEARCH (US) 2019-03-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10220016-B2 Methods and materials for assessing chemotherapy responsiveness and treating cancer PKD2, USP2, BRCA1 MAPT 4230/4885THRB 3869/4885USP2 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.