Metrafenone

Metrafenone

SCHEMBL20788

COc1cc(C)c(C(=O)c2c(OC)ccc(Br)c2C)c(OC)c1OC

nearest known ligand 0.44

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
PTPN1 P18031 2/20 0.40
HTT P42858 2/20 0.39
TSHR P16473 1/20 0.39
APOBEC3A P31941 1/20 0.39
APOBEC3G Q9HC16 1/20 0.39
TUBB1 Q9H4B7 5/20 0.38
HPGD P15428 2/20 0.38
MAPT P10636 2/20 0.38
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
POLB P06746 1/20 0.38
CYP3A4 P08684 1/20 0.38
GFER P55789 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
TUBB4A P04350 3/20 0.38
TUBB P07437 3/20 0.38
TUBA3C P0DPH7 3/20 0.38
TUBA1B P68363 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Metrafenone SCHEMBL30013482 1.00 ALDH1A1 (0.42) ALDH1A1PTPN1HTTTSHRAPOBEC3A
Metrafenone SCHEMBL29408434 1.00 ALDH1A1 (0.42) ALDH1A1PTPN1HTTTSHRAPOBEC3A
SCHEMBL13409130 0.92 ALDH1A1 (0.42) ALDH1A1PTPN1HTTTSHRAPOBEC3A
SCHEMBL6743725 0.92 PTPN1 (0.43) ALDH1A1PTPN1HTTTSHRAPOBEC3A
Metrafenone SCHEMBL1613717 0.92 HPGD (0.52) ALDH1A1TUBB1HPGDMAPTTUBB4A
SCHEMBL6860817 0.91 POLB (0.44) ALDH1A1PTPN1HTTTSHRTUBB1
Metrafenone SCHEMBL2311489 0.91 ALDH1A1 (0.35) ALDH1A1PTPN1HTTTSHRAPOBEC3A
SCHEMBL3762760 0.89 MEN1 (0.39) ALDH1A1PTPN1HTTTSHRAPOBEC3A
SCHEMBL6859535 0.88 ELANE (0.37) ALDH1A1PTPN1HTTTSHRAPOBEC3A
SCHEMBL6699530 0.87 PTPN1 (0.47) ALDH1A1PTPN1HTTTSHRAPOBEC3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 19858 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260137082-A1 FUNGICIDAL COMPOSITIONS COMPRISING FLUDIOXONIL SYNGENTA CROP PROTECTION AG (CH) 2026-05-21 US claimed
WO-2026105160-A1 NOVEL AGROCHEMICAL COMPOSITION COMPRISING 3-SUBSTITUTED PHENYLAMIDINE COMPOUNDS AND USE THEREOF PI INDUSTRIES LTD. (IN) 2026-05-21 WO claimed
WO-2026101908-A1 MIXTURES FOR FUNGAL CONTROL IN SOYBEANS CORTEVA AGRISCIENCE LLC (US) 2026-05-15 WO claimed
WO-2026101906-A1 MIXTURES FOR FUNGAL CONTROL IN CORN CORTEVA AGRISCIENCE LLC (US) 2026-05-15 WO claimed
WO-2026101907-A1 MIXTURES FOR FUNGAL CONTROL IN CEREALS CORTEVA AGRISCIENCE LLC (US) 2026-05-15 WO claimed
WO-2026090564-A2 THIOPHENE BASED APYRASE INHIBITORS TEXAS CROP SCIENCE, INC. (US) 2026-04-30 WO claimed
EP-4447665-B1 FUNGICIDAL COMPOSITIONS SYNGENTA CROP PROTECTION AG (CH) 2026-04-22 EP claimed
EP-4727359-A1 FUNGICIDAL COMPOSITIONS Syngenta Crop Protection AG (CH) 2026-04-22 EP claimed
EP-4710766-A1 MIXTURES OF AMBRUTICIN WITH AT LEAST ONE FURTHER PESTICIDE BASF SE (DE) 2026-03-18 EP claimed
US-20260068884-A1 COMPOSITION USED FOR KILLING FUNGI AND METHOD FOR APPLYING COMPOSITION JIANGSU FLAG CHEMICAL INDUSTRY CO., LTD. (CN) 2026-03-12 US claimed
US-20020065313-A1 Fungicidal mixtures BASF AKTIENGESELLSCHAFT (DE) 2002-05-30 US claimed
EP-1189508-A1 FUNGICIDAL COMPOSITIONS Bayer Aktiengesellschaft (DE) 2002-03-27 EP claimed
EP-1185173-A1 FUNGICIDAL COMBINATIONS Syngenta Participations AG (CH) 2002-03-13 EP claimed
EP-0897904-B1 Fungicidal 2-methoxybenzophenones BASF AG (DE) 2002-02-20 EP claimed
US-6346535-B1 Fungicidal mixtures AMERICAN CYANAMID COMPANY 2002-02-12 US claimed
WO-2001080643-A1 FUNGICIDAL COMPOSITIONS SYNGENTA PARTICIPATIONS AG (CH) 2001-11-01 WO claimed
WO-2000076317-A1 FUNGICIDAL COMBINATIONS SYNGENTA PARTICIPATIONS AG (CH) 2000-12-21 WO claimed
WO-2000072677-A1 FUNGICIDAL COMPOSITIONS BAYER AKTIENGESELLSCHAFT (CH) 2000-12-07 WO claimed
US-5945567-A Fungicidal 2-methoxybenzophenones AMERICAN CYANAMID COMPANY (US) 1999-08-31 US claimed
EP-0897904-A1 Fungicidal 2-methoxybenzophenones American Cyanamid Company (US) 1999-02-24 EP claimed