SCHEMBL20801809

SCHEMBL20801809

CC(C)[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](C)C(=O)Nc1cc2c(c3ccccc13)C(CCl)CN2C(=O)C12CC(C(=O)O)(C1)C2

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 3/20 0.40
PIN1 Q13526 1/20 0.34
ADH1A P07327 1/20 0.33
KIT P10721 1/20 0.33
FLT1 P17948 1/20 0.33
FLT4 P35916 1/20 0.33
KDR P35968 1/20 0.33
ABL2 P42684 1/20 0.33
XIAP P98170 3/20 0.32
EPHX2 P34913 1/20 0.32
BACE1 P56817 1/20 0.32
ELANE P08246 1/20 0.31
MDM4 O15151 1/20 0.31
TP53 P04637 1/20 0.31
FDFT1 P37268 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16933162 1.00 CASP3 (0.40) CASP3PIN1ADH1AKITFLT1
SCHEMBL16933097 0.92 CASP3 (0.37) CASP3PIN1ADH1AKITFLT1
SCHEMBL21297105 0.91 CASP3 (0.39) CASP3PIN1ADH1AKITFLT1
SCHEMBL16933008 0.88 CASP3 (0.35) CASP3PIN1XIAPELANEFDFT1
SCHEMBL16933180 0.88 CASP3 (0.34) CASP3PIN1ADH1AKITFLT1
SCHEMBL16933070 0.86 BACE1 (0.37) CASP3PIN1ADH1AKITFLT1
SCHEMBL21559296 0.86 CASP3 (0.34) CASP3ELANE
SCHEMBL16942085 0.86 CASP3 (0.34) CASP3ELANE
SCHEMBL21234810 0.86 CASP3 (0.38) CASP3PIN1ADH1AKITFLT1
SCHEMBL18064565 0.85 ADH1A (0.38) CASP3PIN1ADH1AKITFLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3521292-A1 BIFUNCTIONAL CYTOTOXIC AGENTS Pfizer Inc (US) 2019-08-07 EP disclosed
EP-3099692-B1 BIFUNCTIONAL CYTOTOXIC AGENTS PFIZER (US) 2019-03-13 EP disclosed