SCHEMBL20802859

SCHEMBL20802859

COC(=O)c1cc(I)c(C)cc1O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 5/20 0.50
CA1 P00915 5/20 0.50
CA2 P00918 5/20 0.50
CA7 P43166 5/20 0.50
CA9 Q16790 5/20 0.50
CA14 Q9ULX7 5/20 0.50
PDK2 Q15119 1/20 0.50
PDK4 Q16654 1/20 0.50
GAA P10253 4/20 0.47
MYC P01106 1/20 0.45
CYP3A4 P08684 2/20 0.44
ACHE P22303 1/20 0.44
LMNA P02545 3/20 0.44
TSHR P16473 1/20 0.44
CFTR P13569 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
HPGD P15428 2/20 0.42
PTGS2 P35354 1/20 0.41
POLB P06746 3/20 0.41
XDH P47989 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1764082 0.85 CA12 (0.46) CA12CA1CA2CA7CA9
SCHEMBL1920431 0.85 CFTR (0.46) CA12CA1CA2CA7CA9
SCHEMBL25455691 0.85 CFTR (0.46) CA12CA1CA2CA7CA9
SCHEMBL30280800 0.85 CFTR (0.46) CA12CA1CA2CA7CA9
SCHEMBL8980551 0.84 CA12 (0.57) CA12CA1CA2CA7CA9
SCHEMBL9128543 0.82 CA12 (0.55) CA12CA1CA2CA7CA9
SCHEMBL27902660 0.82 CA12 (0.55) CA12CA1CA2CA7CA9
SCHEMBL1918973 0.80 GAA (0.50) GAALMNATSHRCFTRSMN1; SMN2
SCHEMBL17239556 0.80 CFTR (0.43) CA12CA1CA2CA7CA9
SCHEMBL19947385 0.80 CFTR (0.46) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019051265-A1 APOPTOSIS SIGNAL-REGULATING KINASE INHIBITORS AND USES THEREOF FRONTHERA U.S. PHARMACEUTICALS LLC (US) 2019-03-14 WO disclosed