SCHEMBL20804359

SCHEMBL20804359

COc1ccc(C(I)c2c(F)ccc(CN3C(=O)C=CC3=O)c2F)cc1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 2/20 0.47
GSK3B P49841 2/20 0.47
MGLL Q99685 1/20 0.35
CMA1 P23946 1/20 0.34
CASP3 P42574 1/20 0.33
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33
NPBWR1 P48145 1/20 0.32
POLB P06746 1/20 0.32
HTT P42858 2/20 0.32
MAPK1 P28482 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
MTNR1B P49286 1/20 0.32
TACR1 P25103 2/20 0.31
ALDH1A1 P00352 1/20 0.31
CHRM1 P11229 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17123212 0.79 GSK3A (0.40) GSK3AGSK3BCASP3HTTMAPK1
SCHEMBL20804233 0.68 MGLL (0.42) GSK3AGSK3BMGLLPTGS1PTGS2
SCHEMBL17123178 0.68 PTGS1 (0.50) GSK3AGSK3BMGLLPTGS1PTGS2
SCHEMBL3384174 0.66 GSK3A (1.00) GSK3AGSK3BMGLLCMA1CASP3
SCHEMBL13486597 0.66 GSK3A (0.58) GSK3AGSK3BPOLBMAPK1ALDH1A1
SCHEMBL11432701 0.63 CA1 (0.58) MAPK1ALDH1A1
SCHEMBL17123192 0.63 GSK3A (0.66) GSK3AGSK3BMGLLCMA1CASP3
SCHEMBL15694366 0.60 GSK3A (0.60) GSK3AGSK3BMGLLCMA1CASP3
SCHEMBL4746479 0.59 KDM4E (0.50) GSK3AGSK3BMGLLPTGS1PTGS2
SCHEMBL3381344 0.58 GSK3A (1.00) GSK3AGSK3BMGLLCMA1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3089962-B1 RADIOIODINATED COMPOUNDS NUTECH VENTURES (US) 2019-03-13 EP disclosed