SCHEMBL20810399

SCHEMBL20810399

C/C=C/c1cnc2ccc(Br)cc2n1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C19 P33261 1/20 0.40
PABPC1 P11940 1/20 0.35
PIK3R1 P27986 1/20 0.34
PIK3CA P42336 1/20 0.34
PAX8 Q06710 1/20 0.34
BACE1 P56817 2/20 0.33
RAB9A P51151 2/20 0.33
EGFR P00533 1/20 0.33
NPC1 O15118 1/20 0.33
ALDH1A1 P00352 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.32
NOS2 P35228 1/20 0.32
PTGES O14684 2/20 0.32
TSHR P16473 1/20 0.31
CASP3 P42574 1/20 0.31
SLC22A12 Q96S37 1/20 0.31
BIRC5 O15392 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12850536 0.79 HTT (0.38) HTTCYP1A2CYP2C19PABPC1PIK3R1
SCHEMBL12850554 0.79 ERN1 (0.39) HTTCYP1A2CYP2C19PABPC1PIK3R1
SCHEMBL2621768 0.79 HTT (0.36) HTTCYP1A2CYP2C19PABPC1PIK3R1
SCHEMBL27127705 0.77 TGFBR1 (0.35) HTTCYP1A2CYP2C19PIK3R1PIK3CA
SCHEMBL29830797 0.77 TGFBR1 (0.35) HTTCYP1A2CYP2C19PIK3R1PIK3CA
SCHEMBL27030609 0.77 TGFBR1 (0.35) HTTCYP1A2CYP2C19PIK3R1PIK3CA
SCHEMBL7940364 0.77 RAB9A (0.50) HTTCYP1A2CYP2C19PAX8RAB9A
SCHEMBL30390906 0.73 HTT (0.41) HTTCYP1A2CYP2C19PABPC1PIK3R1
SCHEMBL1639504 0.73 HTT (0.41) HTTCYP1A2CYP2C19PABPC1PIK3R1
SCHEMBL1758976 0.73 HPGD (0.34) HTTCYP1A2CYP2C19PABPC1PAX8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2916838-B1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS NEUPHARMA INC (US) 2019-03-13 EP disclosed