SCHEMBL20814036

SCHEMBL20814036

Cc1ccc(C=C2C(=O)OC(C)(C)OC2=O)cc1O

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.56
ALDH1A1 P00352 6/20 0.53
CRHBP P24387 1/20 0.53
CRHR2 Q13324 1/20 0.53
SIRT1 Q96EB6 4/20 0.48
LCK P06239 1/20 0.43
MEN1 O00255 4/20 0.42
HPGD P15428 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
ALPL P05186 1/20 0.40
ALPI P09923 1/20 0.40
MAPT P10636 1/20 0.40
ALPG P10696 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
TOP1 P11387 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19551422 0.87 KMT2A (0.59) KMT2AALDH1A1CRHBPCRHR2SIRT1
SCHEMBL16319317 0.81 KMT2A (0.76) KMT2AALDH1A1MEN1ALPLALPI
SCHEMBL435198 0.78 SIRT1 (0.71) KMT2AALDH1A1CRHBPCRHR2SIRT1
SCHEMBL28606256 0.78 KMT2A (0.76) KMT2AALDH1A1SIRT1LCKMEN1
SCHEMBL2497792 0.78 KMT2A (0.59) KMT2AALDH1A1CRHBPCRHR2SIRT1
SCHEMBL17199432 0.76 ALDH1A1 (0.67) KMT2AALDH1A1CRHBPCRHR2SIRT1
SCHEMBL3076148 0.76 KMT2A (0.56) KMT2AALDH1A1CRHBPCRHR2SIRT1
SCHEMBL22409650 0.75 KMT2A (0.56) KMT2AALDH1A1CRHBPCRHR2SIRT1
SCHEMBL12663535 0.75 ALDH1A1 (0.66) KMT2AALDH1A1MEN1CYP1A2CYP3A4
SCHEMBL31462528 0.72 KMT2A (0.56) KMT2AALDH1A1CRHBPCRHR2SIRT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3453704-A1 PHENOL COMPOUND AND COMBINATION OF SAME WITH A BENZODIAZEPINE FUSED TO 1,4-DIHYDROPYRIDINE FOR TREATING DISEASES OF THE CENTRAL NERVOUS AND VASCULAR SYSTEMS Universidad de La Habana (CU) 2019-03-13 EP disclosed