SCHEMBL20814271

SCHEMBL20814271

C[C@H](Oc1ccc(N2CCC3(CCN(CC(O)c4ccc(Cl)cc4Cl)CC3)C3OC32)cn1)C(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
LIPE Q05469 3/20 0.37
KCNH2 Q12809 8/20 0.36
KCNJ1 P48048 8/20 0.36
GRIN2B Q13224 3/20 0.35
ADRA2C P18825 1/20 0.30
TPH1 P17752 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1946323 0.80 LIPE (0.56) CYP3A4CYP2D6CYP2C9CYP2C19LIPE
SCHEMBL1944865 0.80 LIPE (0.56) CYP3A4CYP2D6CYP2C9CYP2C19LIPE
SCHEMBL1943392 0.69 LIPE (0.52) LIPEKCNH2KCNJ1GRIN2B
SCHEMBL1943405 0.69 LIPE (0.52) LIPEKCNH2KCNJ1GRIN2B
SCHEMBL1944403 0.65 LIPE (0.56) LIPEKCNH2KCNJ1
SCHEMBL1947265 0.65 LIPE (0.56) LIPEKCNH2KCNJ1
SCHEMBL12490771 0.61 LIPE (0.43) LIPEKCNH2KCNJ1
SCHEMBL1944235 0.61 LIPE (0.64) LIPEKCNH2KCNJ1
SCHEMBL1944523 0.59 LIPE (0.47) LIPEKCNH2KCNJ1GRIN2B
SCHEMBL5468783 0.59 GRIN2B (0.41) CYP2D6KCNH2KCNJ1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2507239-B1 AZACYCLIC SPIRO DERIVATIVES HOFFMANN LA ROCHE (CH) 2019-03-13 EP disclosed