SCHEMBL20814679

SCHEMBL20814679

O=C1c2ccnc3c(O)ccc(c23)C(=O)N1Cc1ccc(F)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.52
CYP2C19 P33261 1/20 0.52
CASP3 P42574 1/20 0.47
LMNA P02545 3/20 0.46
L3MBTL1 Q9Y468 3/20 0.46
MEN1 O00255 2/20 0.46
RGS12 O14924 2/20 0.46
USP2 O75604 2/20 0.46
MAPT P10636 2/20 0.46
RECQL P46063 2/20 0.46
KMT2A Q03164 2/20 0.46
HTT P42858 1/20 0.46
HPGD P15428 1/20 0.46
UBE2N P61088 1/20 0.46
ATM Q13315 1/20 0.46
CA1 P00915 3/20 0.44
CA2 P00918 3/20 0.44
CA12 O43570 2/20 0.44
CA9 Q16790 2/20 0.44
CYP1B1 Q16678 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20830735 0.88 MEN1 (0.47) CYP1A2CYP2C19LMNAL3MBTL1MEN1
SCHEMBL20830398 0.87 MEN1 (0.46) CYP1A2CYP2C19LMNAL3MBTL1MEN1
SCHEMBL16964861 0.87 CA1 (0.47) CYP1A2CYP2C19LMNAL3MBTL1MEN1
SCHEMBL20830399 0.87 CA12 (0.47) LMNAMEN1RGS12USP2MAPT
SCHEMBL20830748 0.87 MEN1 (0.46) CYP1A2CYP2C19LMNAL3MBTL1MEN1
SCHEMBL16965549 0.87 KMT2A (0.61) CASP3LMNAL3MBTL1MEN1RGS12
SCHEMBL16965144 0.84 KDM4E (0.55) CASP3LMNAMEN1RGS12USP2
SCHEMBL20830510 0.84 APAF1 (0.45) CYP1A2LMNAMEN1RGS12USP2
SCHEMBL16965659 0.84 CLTC (0.43) CYP1A2CYP2C19LMNAL3MBTL1MEN1
SCHEMBL16965485 0.81 CYP1A2 (0.49) CYP1A2CYP2C19CASP3LMNAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2900239-B1 DIHYDRO-6-AZAPHENALENE DERIVATIVES FOR THE TREATMENT OF CNS, OCULAR DISEASES AND RELATED DISORDERS WARNER BABCOCK INST FOR GREEN CHEMISTRY LLC (US) 2019-03-20 EP disclosed
EP-2900239-B1 DIHYDRO-6-AZAPHENALENE DERIVATIVES FOR THE TREATMENT OF CNS, OCULAR DISEASES AND RELATED DISORDERS WARNER BABCOCK INST FOR GREEN CHEMISTRY LLC (US) 2019-03-20 EP disclosed