SCHEMBL20828186

SCHEMBL20828186

CCC[C@@H]1CC[C@H](C(=O)OC)N1C(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.40
CHRM1 P11229 1/20 0.40
CHRM3 P20309 1/20 0.40
ALDH1A1 P00352 3/20 0.36
ATM Q13315 2/20 0.36
KMT2A Q03164 2/20 0.36
CYP3A4 P08684 2/20 0.36
MAPT P10636 2/20 0.36
FKBP1A P62942 1/20 0.36
CETP P11597 1/20 0.34
PREP P48147 3/20 0.34
PTPN1 P18031 1/20 0.34
EPHX1 P07099 1/20 0.33
NR1H2 P55055 2/20 0.32
NR1H3 Q13133 1/20 0.32
GPR119 Q8TDV5 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
MEN1 O00255 1/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30642071 1.00 CHRM2 (0.40) CHRM2CHRM1CHRM3ALDH1A1ATM
SCHEMBL22454897 0.92 FKBP1A (0.42) CHRM2CHRM1CHRM3ALDH1A1ATM
SCHEMBL22454898 0.92 FKBP1A (0.42) CHRM2CHRM1CHRM3ALDH1A1ATM
SCHEMBL30918110 0.89 CHRM2 (0.40) CHRM2CHRM1CHRM3ALDH1A1FKBP1A
SCHEMBL27380504 0.89 CHRM2 (0.40) CHRM2CHRM1CHRM3ALDH1A1FKBP1A
SCHEMBL24894588 0.89 CHRM2 (0.40) CHRM2CHRM1CHRM3ALDH1A1FKBP1A
SCHEMBL24894365 0.89 CHRM2 (0.40) CHRM2CHRM1CHRM3ALDH1A1FKBP1A
SCHEMBL5368239 0.89 CHRM2 (0.42) CHRM2CHRM1CHRM3ALDH1A1KMT2A
SCHEMBL18430796 0.88 CHRM2 (0.39) CHRM2CHRM1CHRM3ALDH1A1ATM
SCHEMBL24894638 0.86 CHRM2 (0.38) CHRM2CHRM1CHRM3ALDH1A1FKBP1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12378216-B2 Heteroaryl(heterocyclyl)methanol compounds useful in the treatment of hyperglycaemia ATROGI AB (SE) 2025-08-05 US disclosed
EP-3681862-B1 BETA-HYDROXY HETEROCYCLIC AMINES AND THEIR USE IN THE TREATMENT OF HYPERGLYCAEMIA ATROGI AB (SE) 2023-11-08 EP disclosed
US-11427539-B2 Beta-hydroxy heterocyclic amines and their use in the treatment of hyperglycaemia ATROGI AB (SE) 2022-08-30 US disclosed
US-20220194920-A1 HETEROARYL(HETEROCYCLYL)METHANOL COMPOUNDS USEFUL IN THE TREATMENT OF HYPERGLYCAEMIA ATROGI AB (SE) 2022-06-23 US disclosed
US-20220194920-A1 HETEROARYL(HETEROCYCLYL)METHANOL COMPOUNDS USEFUL IN THE TREATMENT OF HYPERGLYCAEMIA ATROGI AB (SE) 2022-06-23 US disclosed
CN-113784961-A Heteroaryl (heterocyclyl) carbinol compounds useful for treating hyperglycemia 阿托基公司 2021-12-10 CN disclosed
US-20200277259-A1 BETA-HYDROXY HETEROCYCLIC AMINES AND THEIR USE IN THE TREATMENT OF HYPERGLYCAEMIA ATROGI AB (SE) 2020-09-03 US disclosed
WO-2019053425-A1 BETA-HYDROXY HETEROCYCLIC AMINES AND THEIR USE IN THE TREATMENT OF HYPERGLYCAEMIA ATROGI AB (SE) 2019-03-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200277259-A1 BETA-HYDROXY HETEROCYCLIC AMINES AND THEIR USE IN THE TREATMENT OF HYPERGLYCAEMIA SLC5A1, GPR119, SLC5A2 CHRM2 756/4885CHRM1 314/4885CHRM3 1396/4885
US-11427539-B2 Beta-hydroxy heterocyclic amines and their use in the treatment of hyperglycaemia SLC5A1, GPR119, SLC5A2 CHRM2 756/4885CHRM1 314/4885CHRM3 1396/4885
US-12378216-B2 Heteroaryl(heterocyclyl)methanol compounds useful in the treatment of hyperglycaemia SLC5A1, GPR119, SLC5A2 CHRM2 353/4885CHRM1 145/4885CHRM3 855/4885
US-20220194920-A1 HETEROARYL(HETEROCYCLYL)METHANOL COMPOUNDS USEFUL IN THE TREATMENT OF HYPERGLYCAEMIA SLC5A1, GPR119, SLC5A2 CHRM2 353/4885CHRM1 145/4885CHRM3 855/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.