SCHEMBL20834898

SCHEMBL20834898

CCc1cc(C)ccc1C#Cc1cc(F)c(N)c(F)c1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 10/20 0.36
FFAR4 Q5NUL3 6/20 0.36
TAAR1 Q96RJ0 1/20 0.33
GRM4 Q14833 1/20 0.32
HSP90B1 P14625 1/20 0.32
TRAP1 Q12931 1/20 0.32
ACACB O00763 1/20 0.31
CA12 O43570 1/20 0.31
CA2 P00918 1/20 0.31
CA9 Q16790 1/20 0.31
NOS3 P29474 1/20 0.30
NOS1 P29475 1/20 0.30
NOS2 P35228 1/20 0.30
TSPO P30536 1/20 0.30
DRD3 P35462 1/20 0.30
KDR P35968 2/20 0.30
PDGFRB P09619 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30462077 0.84 ACACB (0.39) FFAR1FFAR4HSP90B1TRAP1ACACB
SCHEMBL20819526 0.84 ACACB (0.39) FFAR1FFAR4HSP90B1TRAP1ACACB
SCHEMBL23309992 0.82 FFAR1 (0.46) FFAR1FFAR4GRM4CA12CA2
SCHEMBL21396283 0.80 GABRA1 (0.41) FFAR1FFAR4TSPODRD3
SCHEMBL20834872 0.80 FFAR1 (0.34) FFAR1FFAR4TSPODRD3
SCHEMBL20819525 0.79 HTR2A (0.38) FFAR1FFAR4CA2
SCHEMBL30462104 0.79 HTR2A (0.38) FFAR1FFAR4CA2
SCHEMBL19412665 0.76 FFAR1 (0.32) FFAR1FFAR4
SCHEMBL7851688 0.73 FFAR1 (0.47) FFAR1FFAR4ACACBTSPODRD3
SCHEMBL20118652 0.72 FFAR1 (0.40) FFAR1FFAR4ACACBCA12CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3681976-B1 ISOTHIOCYANATO TOLANE DERIVATIVES MERCK PATENT GMBH (DE) 2021-05-26 EP disclosed
WO-2019052972-A1 ISOTHIOCYANATO TOLANE DERIVATIVES MERCK PATENT GMBH (DE) 2019-03-21 WO disclosed