SCHEMBL20840671

SCHEMBL20840671

CCOC(=O)CCc1cccc(NC(=O)c2ccccc2NC(=O)c2ccc(-n3ccnn3)cc2)c1

nearest known ligand 0.54

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 12/20 0.54
PPARG P37231 8/20 0.54
PPARA Q07869 8/20 0.54
PPARD Q03181 10/20 0.51
ABCG2 Q9UNQ0 2/20 0.45
F10 P00742 2/20 0.44
RXFP1 Q9HBX9 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
HSPH1 Q92598 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20852078 0.88 NR1H4 (0.66) NR1H4PPARGPPARAPPARDF10
SCHEMBL20840670 0.84 MAPK9 (0.47)
SCHEMBL20839629 0.79 NR1H4 (0.56) NR1H4PPARGPPARAPPARDABCG2
SCHEMBL20839777 0.79 NR1H4 (0.56) NR1H4PPARGPPARAPPARDABCG2
SCHEMBL20839957 0.78 NR1H4 (0.58) NR1H4PPARGPPARAPPARDABCG2
SCHEMBL20839668 0.78 NR1H4 (0.56) NR1H4PPARGPPARAPPARDABCG2
SCHEMBL20839618 0.78 NR1H4 (0.53) NR1H4PPARGPPARAPPARDABCG2
SCHEMBL20839596 0.78 NR1H4 (0.57) NR1H4PPARGPPARAPPARDABCG2
SCHEMBL20839724 0.77 CYP3A4 (0.52) NR1H4PPARGPPARAPPARDABCG2
SCHEMBL7043921 0.77 NOTUM (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019057969-A1 DUAL AGONISTS OF FXR AND PPARδ AND THEIR USES Johann Wolfgang Goethe-Universität (DE) 2019-03-28 WO disclosed